Target Details
| UniProt AC | O15146 |
|---|---|
| Gene Symbol | MUSK |
| Protein Name | Muscle, skeletal receptor tyrosine-protein kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01392 (Fz) PF07679 (I-set) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 29
- Clinical molecules 7
- Avg pChEMBL 6.79
Associated Diseases (2)
Active Molecules (29)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ODPGGGTTYSGTGO
|
8.5 | Kd | 153 | — | |
MPVGZUGXCQEXTM
|
8.0 | Kd | 61 | Yes | |
CXQHYVUVSFXTMY
|
7.9 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
7.9 | Kd | 149 | — | |
YOBIWCLAYQWPPW
|
7.9 | IC50 | 23 | — | |
BPIWZDNVMQQBQX
|
7.3 | IC50 | 5 | — | |
HKSZLNNOFSGOKW
|
7.1 | IC50 | 408 | — | |
HKSZLNNOFSGOKW
|
7.1 | Kd | 213 | — | |
CTNPALGJUAXMMC
|
7.0 | Kd | 151 | — | |
NHHQJBCNYHBUSI
|
7.0 | Kd | 220 | — | |
ZHOXAGNPCZTRBN
|
7.0 | Kd | 20 | — | |
MLDQJTXFUGDVEO
|
6.9 | Kd | 85 | Yes | |
YYLKKYCXAOBSRM
|
6.7 | Kd | 191 | — | |
HIHOEGPXVVKJPP
|
6.7 | IC50 | 10 | — | |
KTEIFNKAUNYNJU
|
6.6 | Kd | 114 | — | |
YLCFOHVAOBLAIK
|
6.6 | IC50 | 14 | — | |
QQWUGDVOUVUTOY
|
6.6 | Kd | 231 | Yes | |
GCIKSSRWRFVXBI
|
6.5 | Kd | 109 | Yes | |
LJODJUIHONTDMR
|
6.5 | IC50 | 7 | — | |
WINHZLLDWRZWRT
|
6.3 | Kd | 201 | Yes | |
CMJJZRAAQMUAFH
|
6.3 | Kd | 9 | — | |
XZXHXSATPCNXJR
|
6.2 | Kd | 165 | Yes | |
DUKJABPGWUISRC
|
6.2 | IC50 | 10 | — | |
JOOXLOJCABQBSG
|
6.1 | Kd | 139 | — | |
PIQCTGMSNWUMAF
|
6.1 | Kd | 137 | Yes | |
CVWXJKQAOSCOAB
|
6.0 | Kd | 35 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |