Target Details
| UniProt AC | O15075 |
|---|---|
| Gene Symbol | DCLK1 |
| Protein Name | Serine/threonine-protein kinase DCLK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF03607 (DCX) PF00069 (Pkinase) |
Summary
- Multi-target molecules 44
- Clinical molecules 3
- Avg pChEMBL 7.15
Active Molecules (44)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QRVNXVTYIYXPER
|
9.0 | IC50 | 3 | — | |
DDJBEYRDSUCNLT
|
8.7 | IC50 | 4 | — | |
ISCJKSNXTHTNBW
|
8.5 | IC50 | 4 | — | |
REPCEIPSIPNRSG
|
8.5 | IC50 | 3 | — | |
DDTPGANIPBKTNU
|
8.4 | IC50 | 8 | — | |
JVSJTGAAAMSIAW
|
8.4 | IC50 | 2 | — | |
QQWUGDVOUVUTOY
|
8.3 | Kd | 231 | Yes | |
WVDQWAPBMCRMGM
|
8.0 | IC50 | 2 | — | |
WUWXJIFZTHONGM
|
8.0 | IC50 | 3 | — | |
NGSRRJBACKDZHY
|
7.8 | IC50 | 3 | — | |
XVBGRTMNFNMINE
|
7.7 | IC50 | 5 | — | |
NFNBVXVXMQZSGB
|
7.6 | IC50 | 3 | — | |
YRDHKIFCGOZTGD
|
7.6 | IC50 | 21 | — | |
WWDLVMCJDNTBPK
|
7.5 | IC50 | 3 | — | |
JVVFSGBLMWRDED
|
7.4 | IC50 | 2 | — | |
XKFTZKGMDDZMJI
|
7.4 | Ki | 56 | — | |
HGHFBVBNHYJNHK
|
7.3 | IC50 | 3 | — | |
GBGQVKUZCXSIOV
|
7.2 | IC50 | 2 | — | |
LIEUQFMVFKJKHX
|
7.2 | Kd | 10 | — | |
HFNKQEVNSGCOJV
|
7.2 | Kd | 65 | — | |
YYTFTZONXCQXLW
|
7.2 | IC50 | 3 | — | |
YSFFGUHMDPYPAW
|
7.0 | IC50 | 3 | — | |
DWHWHOPFYUJPCQ
|
7.0 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.0 | Kd | 213 | — | |
KCMYPBPMTXEKNF
|
7.0 | IC50 | 7 | — | |
OWRXHGAFWZFFCW
|
6.9 | Ki | 113 | — | |
ZQUIUVSYHRHZHW
|
6.9 | IC50 | 2 | — | |
JGVXSQJYBQAPAE
|
6.8 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
6.8 | IC50 | 408 | — | |
CRFHZXHUGPCWJA
|
6.7 | IC50 | 8 | — | |
JOOXLOJCABQBSG
|
6.7 | Kd | 139 | — | |
MMMPFWNSQKXKDX
|
6.5 | Ki | 14 | — | |
KTEIFNKAUNYNJU
|
6.5 | Kd | 114 | — | |
WINHZLLDWRZWRT
|
6.4 | Kd | 201 | Yes | |
NPRYKZQCTXZUKH
|
6.3 | IC50 | 2 | — | |
XZXHXSATPCNXJR
|
6.3 | Kd | 165 | Yes | |
CTNPALGJUAXMMC
|
6.3 | Kd | 151 | — | |
GCYXEGSPUDSZJY
|
6.2 | Ki | 82 | — | |
UNVKXVCDLOLPJE
|
6.2 | Ki | 8 | — | |
MVJMMLFMPWITEJ
|
6.1 | Ki | 110 | — | |
UMTWTCVTRDYHQQ
|
6.1 | Ki | 56 | — | |
ADMFLILDQJSEIK
|
6.0 | Ki | 72 | — | |
BSFNGHCTZDCQBF
|
6.0 | Ki | 93 | — | |
RIBBPSYZBQQTQC
|
6.0 | Ki | 15 | — |