Target Details
| UniProt AC | O15047 |
|---|---|
| Gene Symbol | SETD1A |
| Protein Name | Histone-lysine N-methyltransferase SETD1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF11764 (N-SET) PF00076 (RRM_1) PF00856 (SET) |
Summary
- Multi-target molecules 1
- Clinical molecules 0
- Avg pChEMBL 7.29
KEGG Pathways (2)
Associated Diseases (2)
Active Molecules (1)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AAAQFGUYHFJNHI
|
7.3 | IC50 | 252 | — |