Target Details
| UniProt AC | O14976 |
|---|---|
| Gene Symbol | GAK |
| Protein Name | Cyclin-G-associated kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF10409 (PTEN_C2) |
Summary
- Multi-target molecules 134
- Clinical molecules 31
- Avg pChEMBL 6.97
Active Molecules (134)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IVRXNBXKWIJUQB
|
6.3 | Kd | 10 | — | |
NTOMZGNNDKIPEH
|
6.3 | Ki | 4 | — | |
CJIAUJUVHMAHQC
|
6.2 | Ki | 4 | — | |
YBXRSCXGRPSTMW
|
6.2 | Kd | 6 | — | |
IJDQETGUEUJVTB
|
6.2 | Kd | 4 | — | |
HVXKQKFEHMGHSL
|
6.2 | Kd | 21 | — | |
RHXHGRAEPCAFML
|
6.2 | Kd | 9 | — | |
HWXVIOGONBBTBY
|
6.2 | Kd | 27 | — | |
KKKRKRMVJRHDMG
|
6.2 | Kd | 14 | — | |
GOOYSJIWTIHOGW
|
6.1 | IC50 | 3 | — | |
QQLKULDARVNMAL
|
6.1 | Kd | 4 | — | |
MCYCSSJHDPRHBZ
|
6.1 | Ki | 4 | — | |
RKAHOQATMSONTM
|
6.1 | IC50 | 6 | — | |
JMGXJHWTVBGOKG
|
6.1 | Kd | 7 | — | |
GUBJNPWVIUFSTR
|
6.1 | Kd | 103 | — | |
USXZHEGWWNBLBI
|
6.1 | Ki | 4 | — | |
BPYJNSODEPCDRH
|
6.0 | IC50 | 2 | — | |
CWDJCUXKEDKAQE
|
6.0 | IC50 | 2 | — | |
GGYXFRIDIFIYBO
|
6.0 | IC50 | 2 | — | |
GTQNBLFIFRGIBF
|
6.0 | IC50 | 2 | — | |
HNPFCASNBZNQNU
|
6.0 | IC50 | 2 | — | |
HQMHIXREFMNYET
|
6.0 | IC50 | 2 | — | |
HXRGDEBGHHKEEK
|
6.0 | IC50 | 2 | — | |
IBPRZGYJJMUZLP
|
6.0 | IC50 | 2 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KTUFNOKKBVMGRW
|
6.0 | Kd | 38 | Yes | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MHWJYODTCNDXJW
|
6.0 | IC50 | 2 | — | |
NSQIWTMRSLRZLP
|
6.0 | IC50 | 2 | — | |
OVOUHRFMZBHNMX
|
6.0 | IC50 | 2 | — | |
RETYBSQLAYVBLT
|
6.0 | IC50 | 2 | — | |
RJNDAWMSDOWAKQ
|
6.0 | IC50 | 2 | — | |
STOKTXVQCBDPNW
|
6.0 | IC50 | 2 | — |