Target Details
| UniProt AC | O14976 |
|---|---|
| Gene Symbol | GAK |
| Protein Name | Cyclin-G-associated kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF10409 (PTEN_C2) |
Summary
- Multi-target molecules 134
- Clinical molecules 31
- Avg pChEMBL 6.97
Active Molecules (134)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JKCNRFQYOHWEDM
|
7.0 | IC50 | 2 | — | |
JKCNRFQYOHWEDM
|
7.0 | IC50 | 2 | — | |
NSQIWTMRSLRZLP
|
7.0 | IC50 | 2 | — | |
OMZCMEYTWSXEPZ
|
7.0 | Kd | 43 | Yes | |
WSEPAQYPZMEAQP
|
7.0 | IC50 | 2 | — | |
OUKYUETWWIPKQR
|
7.0 | Kd | 31 | Yes | |
AWSQADBSXFTFKL
|
7.0 | Kd | 5 | — | |
JXDYOSVKVSQGJM
|
6.9 | Kd | 7 | — | |
XUZMWHLSFXCVMG
|
6.9 | Kd | 24 | — | |
BOOFYGICEYSNIB
|
6.8 | Kd | 2 | — | |
IBGLGMOPHJQDJB
|
6.8 | Kd | 8 | Yes | |
SVNVPNHWFJFRLZ
|
6.8 | IC50 | 8 | — | |
LVXJQMNHJWSHET
|
6.8 | Kd | 7 | — | |
DFJSJLGUIXFDJP
|
6.8 | Kd | 9 | — | |
BPNUQXPIQBZCMR
|
6.7 | Kd | 83 | Yes | |
XQVVPGYIWAGRNI
|
6.7 | Kd | 34 | — | |
CUIHSIWYWATEQL
|
6.7 | Kd | 61 | Yes | |
IAYGCINLNONXHY
|
6.7 | Kd | 50 | — | |
HINOQCZIDBNXEI
|
6.7 | IC50 | 5 | — | |
XLOGLWKOHPIJLV
|
6.7 | Ki | 3 | — | |
IYHHRZBKXXKDDY
|
6.7 | IC50 | 6 | — | |
JWNPDZNEKVCWMY
|
6.6 | Kd | 57 | Yes | |
NHHQJBCNYHBUSI
|
6.6 | Kd | 220 | — | |
KDGFLJKFZUIJMX
|
6.6 | Kd | 10 | — | |
YYLKKYCXAOBSRM
|
6.6 | Kd | 191 | — | |
HZTYDQRUAWIZRE
|
6.6 | Kd | 40 | Yes | |
MFAQYJIYDMLAIM
|
6.5 | Kd | 130 | Yes | |
JAWYVNPEVKLENS
|
6.5 | IC50 | 2 | — | |
JKCNRFQYOHWEDM
|
6.5 | IC50 | 2 | — | |
NSQIWTMRSLRZLP
|
6.5 | IC50 | 2 | — | |
NTXHJAVJAVSTET
|
6.5 | IC50 | 2 | — | |
OVUOFYVATYZDTQ
|
6.5 | IC50 | 2 | — | |
WSEPAQYPZMEAQP
|
6.5 | IC50 | 2 | — | |
ZZVWLSVVRDNANL
|
6.5 | IC50 | 2 | — | |
WCVTXEYTMLUPPQ
|
6.5 | IC50 | 2 | — | |
QKAONCSNINNEGU
|
6.4 | Kd | 5 | — | |
YSMDVXCUNQWGNN
|
6.4 | Ki | 4 | — | |
BIIVYFLTOXDAOV
|
6.4 | Kd | 29 | — | |
BIIVYFLTOXDAOV
|
6.4 | Kd | 82 | Yes | |
BMGQWWVMWDBQGC
|
6.4 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.4 | Kd | 91 | Yes | |
HVHRHDHQHUAOQI
|
6.4 | IC50 | 5 | — | |
RGZXAQQHXALOBL
|
6.4 | Kd | 10 | — | |
ZZSBPGIGIUFJRA
|
6.4 | Kd | 46 | — | |
FFTUIKFDUYMWTI
|
6.4 | IC50 | 5 | — | |
XCOSAQGGGZDYJN
|
6.4 | Kd | 11 | — | |
DDTPGANIPBKTNU
|
6.3 | Kd | 8 | — | |
HUFOZJXAKZVRNJ
|
6.3 | Kd | 10 | — | |
PLIVFNIUGLLCEK
|
6.3 | Kd | 20 | Yes | |
PIQCTGMSNWUMAF
|
6.3 | Kd | 137 | Yes |