Target Details
| UniProt AC | O14976 |
|---|---|
| Gene Symbol | GAK |
| Protein Name | Cyclin-G-associated kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF10409 (PTEN_C2) |
Summary
- Multi-target molecules 134
- Clinical molecules 31
- Avg pChEMBL 6.97
Active Molecules (134)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CSGQVNMSRKWUSH
|
9.5 | Kd | 21 | — | |
KTSDBMVHAKWDRK
|
9.3 | IC50 | 2 | — | |
LNRFTLQUUQAWMM
|
9.0 | IC50 | 4 | Yes | |
JOOXLOJCABQBSG
|
9.0 | Kd | 139 | — | |
UBPYILGKFZZVDX
|
8.9 | Kd | 130 | Yes | |
AQSSMEORRLJZLU
|
8.7 | Kd | 34 | Yes | |
ZBNZXTGUTAYRHI
|
8.6 | Kd | 102 | Yes | |
AAKJLRGGTJKAMG
|
8.5 | Kd | 50 | Yes | |
XLSYZSRXVVCHLS
|
8.4 | Kd | 48 | — | |
AHESYZXOYPHUOT
|
8.4 | Kd | 4 | — | |
AUOSKLDNVNGKRR
|
8.3 | IC50 | 6 | — | |
DKZYXHCYPUVGAF
|
8.3 | Kd | 112 | — | |
FCDUXQUQGSKWMD
|
8.3 | Kd | 2 | — | |
QQWUGDVOUVUTOY
|
8.3 | Kd | 231 | Yes | |
ULCIVHLQFMURQB
|
8.2 | Kd | 2 | — | |
WVUNYSQLFKLYNI
|
8.2 | Kd | 46 | Yes | |
FQUBTLMSWPIBBP
|
8.2 | Kd | 4 | — | |
UIARLYUEJFELEN
|
8.1 | Kd | 289 | Yes | |
QPDPAWXTOAVKLC
|
8.1 | Kd | 2 | — | |
VAARYSWULJUGST
|
8.1 | Kd | 119 | Yes | |
YULUHUJTIHWRMI
|
8.1 | Kd | 4 | — | |
JONPTLGCLPUHKH
|
8.1 | Kd | 8 | — | |
AAUCXXCMBFZYRT
|
8.1 | Kd | 2 | — | |
ILBOKEFXMPHJKP
|
8.1 | IC50 | 2 | — | |
XGALLCVXEZPNRQ
|
7.9 | Kd | 39 | Yes | |
KRAYLQVJPUMBPE
|
7.8 | Kd | 2 | — | |
VYPGLYMWNDRFGZ
|
7.8 | IC50 | 12 | — | |
HKSZLNNOFSGOKW
|
7.8 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
7.8 | Kd | 213 | — | |
WINHZLLDWRZWRT
|
7.7 | Kd | 201 | Yes | |
BLWQIEISIMYCHD
|
7.7 | Kd | 4 | — | |
XOTGKYTUNDYTBS
|
7.7 | IC50 | 3 | — | |
YFNWWNRZJGMDBR
|
7.6 | Kd | 35 | — | |
GRKVQPWSPUXGKV
|
7.6 | Kd | 3 | — | |
FPWOHBGDJPLADA
|
7.5 | Kd | 4 | — | |
ZUNCPEIOPMEIGV
|
7.5 | Kd | 4 | — | |
FKLSPSFZXNNVKC
|
7.5 | Kd | 2 | — | |
KRIUNPBAQZGFQA
|
7.4 | Kd | 76 | — | |
CDMGBJANTYXAIV
|
7.4 | Kd | 34 | Yes | |
CQKFTSMPIIYOBX
|
7.4 | IC50 | 3 | Yes | |
CTNPALGJUAXMMC
|
7.4 | Kd | 151 | — | |
QHKYPYXTTXKZST
|
7.3 | Kd | 28 | — | |
RNCVPFCGSMNPPO
|
7.2 | IC50 | 5 | Yes | |
WMAOMQUWVSXRPR
|
7.2 | IC50 | 2 | — | |
NGBWQVJCOYTGOR
|
7.1 | IC50 | 8 | — | |
ULXXDDBFHOBEHA
|
7.1 | Kd | 15 | Yes | |
UHTHHESEBZOYNR
|
7.1 | Kd | 66 | Yes | |
LSPANGZZENHZNJ
|
7.1 | IC50 | 10 | Yes | |
ITTRLTNMFYIYPA
|
7.0 | Kd | 17 | — | |
HFNKQEVNSGCOJV
|
7.0 | Kd | 65 | — |