Target Details
| UniProt AC | O14965 |
|---|---|
| Gene Symbol | AURKA |
| Protein Name | Aurora kinase A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,119
- Clinical molecules 389
- Avg pChEMBL 7.5
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (2,119)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GUKUYYRQJNMIEZ
|
8.6 | Kd | 2 | — | |
HOPYTUITHBXQSC
|
8.6 | IC50 | 5 | Yes | |
WHOKGFKDKLABFY
|
8.6 | IC50 | 2 | — | |
WHOKGFKDKLABFY
|
8.6 | IC50 | 2 | — | |
JGBVPRGLWQWHIG
|
8.5 | IC50 | 2 | — | |
KXICNNJQUUCJQT
|
8.5 | IC50 | 3 | — | |
QWMDXMFYSJOKEB
|
8.5 | IC50 | 2 | — | |
GEATXDJAPAHPTP
|
8.5 | IC50 | 10 | — | |
KPCFWSWNBPMJIY
|
8.5 | IC50 | 2 | — | |
LDWBULFGVRAVMR
|
8.5 | Ki | 3 | — | |
LNGVCHKMQJKHDR
|
8.5 | Ki | 6 | Yes | |
LYDTZBUSUCDSRL
|
8.5 | IC50 | 3 | Yes | |
MBKBRIBQHFBRHO
|
8.5 | IC50 | 3 | — | |
NGEVHWVGFQLFEK
|
8.5 | IC50 | 3 | — | |
PEPCSEJJADXCRB
|
8.5 | Ki | 4 | Yes | |
PEXOYGNRWYUDOM
|
8.5 | IC50 | 3 | — | |
SVXYIHAHZMQVBU
|
8.5 | IC50 | 2 | — | |
UANPKXDLMMRBAX
|
8.5 | IC50 | 2 | — | |
YQQWGLNBSUZDRG
|
8.5 | IC50 | 2 | — | |
YUAALFPUEOYPNX
|
8.5 | IC50 | 3 | — | |
ZLODPJRHCQWJSX
|
8.5 | IC50 | 3 | — | |
ALKJNCZNEOTEMP
|
8.5 | IC50 | 55 | — | |
GADYBZMYJCZJLX
|
8.5 | IC50 | 2 | — | |
GWQXSFUEKBLIOK
|
8.5 | IC50 | 3 | — | |
MLRUASYAPWIQDS
|
8.5 | IC50 | 2 | — | |
PZRFGYNACSHNJL
|
8.5 | IC50 | 2 | — | |
SSJZAOVCTAZHIR
|
8.5 | IC50 | 3 | — | |
BIKYDWLMTPRSQL
|
8.5 | Ki | 50 | — | |
KNARVZUUCLIBGV
|
8.5 | Ki | 33 | — | |
ZJQWORQRPDYKRS
|
8.5 | IC50 | 7 | — | |
FGKOFCQQLIEQOZ
|
8.5 | IC50 | 2 | — | |
HOYCAZAYAZDSGA
|
8.5 | IC50 | 2 | — | |
AKSIZPIFQAYJGF
|
8.5 | IC50 | 4 | Yes | |
BJLXYCDZTRNOAH
|
8.5 | IC50 | 3 | — | |
PRBRXSXEFQRILZ
|
8.5 | IC50 | 2 | — | |
ZCNHSWBTKSJQNS
|
8.5 | IC50 | 3 | — | |
CMEKRUHUVGTVLK
|
8.5 | IC50 | 6 | Yes | |
MNYJXBQMADDOQS
|
8.5 | IC50 | 3 | — | |
ZQCJERNZTUANGM
|
8.5 | IC50 | 3 | — | |
BZJOCZCFTSVKLT
|
8.4 | IC50 | 2 | — | |
BZJOCZCFTSVKLT
|
8.4 | IC50 | 2 | — | |
OQAVDYCSFNEKFW
|
8.4 | IC50 | 2 | — | |
PZRFGYNACSHNJL
|
8.4 | IC50 | 2 | — | |
BRVRJAZHVITNIF
|
8.4 | IC50 | 3 | Yes | |
PHENCDSAYZNXRO
|
8.4 | IC50 | 3 | — | |
RLEBVXHKDJKLHD
|
8.4 | IC50 | 2 | — | |
AGHMFEHJWZVACU
|
8.4 | Ki | 3 | Yes | |
BXFVYQXRSWCGMU
|
8.4 | IC50 | 3 | — | |
GBXVVXZXFOFHSU
|
8.4 | Ki | 3 | Yes | |
NHNIQMDXSHWKPU
|
8.4 | IC50 | 2 | — |