Target Details
| UniProt AC | O14965 |
|---|---|
| Gene Symbol | AURKA |
| Protein Name | Aurora kinase A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,119
- Clinical molecules 389
- Avg pChEMBL 7.5
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (2,119)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BPQKNCMYCHBDMJ
|
8.7 | IC50 | 2 | — | |
BRTHUECZMVKNMQ
|
8.7 | Ki | 31 | — | |
DYAYBUDFGBTDNI
|
8.7 | IC50 | 2 | Yes | |
HCDXOVUMIOIELK
|
8.7 | IC50 | 3 | — | |
HWUIJIOSFJIUGC
|
8.7 | Ki | 2 | — | |
IDOIWFPLBQQGRQ
|
8.7 | IC50 | 3 | — | |
KLZCFIRMAFXIKI
|
8.7 | IC50 | 3 | — | |
LLSACPYCBRAUIJ
|
8.7 | IC50 | 2 | — | |
OSZWVKNIHJPNFJ
|
8.7 | IC50 | 2 | — | |
OWFXKTOLFUQPDJ
|
8.7 | Ki | 36 | — | |
PSWIPMICOQJHRP
|
8.7 | IC50 | 3 | — | |
RQNRFNOSAPOJTQ
|
8.7 | IC50 | 2 | — | |
SYZBPKURKLVKGY
|
8.7 | IC50 | 3 | — | |
UAZXSLJQCXJPNG
|
8.7 | Ki | 2 | — | |
VKXOHXJUQSDMJO
|
8.7 | IC50 | 2 | — | |
VMAMZHADUWRQFW
|
8.7 | IC50 | 3 | — | |
WKKLEERAKHQFTN
|
8.7 | IC50 | 3 | — | |
XHORJSJFHVABEA
|
8.7 | Ki | 49 | — | |
XUAORJVHYWCADO
|
8.7 | Ki | 5 | Yes | |
ZGCQIBQYASDQPM
|
8.7 | IC50 | 3 | — | |
ZNZJOKVVRNTGRH
|
8.7 | IC50 | 2 | — | |
KCMYPBPMTXEKNF
|
8.7 | IC50 | 7 | — | |
BRXIQCXGFZUJEE
|
8.7 | IC50 | 3 | — | |
BTZLYPOEWBMAMN
|
8.7 | IC50 | 2 | — | |
VMAAFUOXTWPYRN
|
8.7 | IC50 | 9 | Yes | |
NUAVXRQHCVNICO
|
8.7 | IC50 | 2 | — | |
WWPXOBSLFBHGEZ
|
8.7 | IC50 | 3 | — | |
BPXZXMRLFSWKLW
|
8.6 | IC50 | 3 | — | |
DZJJTOUVFUJWPC
|
8.6 | IC50 | 2 | — | |
KXEJAEQUXNWZTK
|
8.6 | IC50 | 2 | — | |
MFRRIEBIBJQMAF
|
8.6 | IC50 | 3 | — | |
SCBRGKRRYRGFMN
|
8.6 | IC50 | 2 | — | |
SDEWZAPYGJGVJM
|
8.6 | IC50 | 2 | — | |
URHJZIHVIAKFBP
|
8.6 | IC50 | 2 | — | |
YCKYDQJFSLJBKW
|
8.6 | IC50 | 2 | — | |
GJDYHJPLCHRKEK
|
8.6 | IC50 | 3 | — | |
KAQWYRBKYUAJGJ
|
8.6 | IC50 | 2 | — | |
LEWVUPUKJSFGLR
|
8.6 | Ki | 3 | Yes | |
UYNUFNIQHUWLML
|
8.6 | IC50 | 2 | — | |
ZUOHNZIRNKHHJE
|
8.6 | Ki | 3 | Yes | |
HKSZLNNOFSGOKW
|
8.6 | Ki | 118 | — | |
IAKGNUWZPSPEKU
|
8.6 | Ki | 19 | — | |
RZRPIHMYICQRMC
|
8.6 | IC50 | 2 | — | |
VBXXGYSKTLTOBL
|
8.6 | Kd | 2 | — | |
ZZCZGLYROGNMLJ
|
8.6 | IC50 | 3 | — | |
BZUCVINJZSBGPK
|
8.6 | IC50 | 3 | — | |
GZZPKHLUNHCCCE
|
8.6 | IC50 | 3 | — | |
RWCPLVNQNAADEI
|
8.6 | IC50 | 2 | — | |
LNSIQBCMRAUWIA
|
8.6 | IC50 | 2 | — | |
UWVYYAZEVUASFC
|
8.6 | IC50 | 3 | — |