Target Details
| UniProt AC | O14965 |
|---|---|
| Gene Symbol | AURKA |
| Protein Name | Aurora kinase A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,119
- Clinical molecules 389
- Avg pChEMBL 7.5
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (2,119)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SEYBQYNGNHTWDW
|
9.0 | IC50 | 2 | — | |
URYOYOMAOIZWMC
|
9.0 | IC50 | 2 | — | |
UUQUQPUHXKTHDD
|
9.0 | IC50 | 2 | — | |
YEDBJKRVUNJEML
|
9.0 | IC50 | 3 | — | |
JGFQBBRDUAPPHV
|
8.9 | IC50 | 2 | — | |
JMLSGXAFWBMOHG
|
8.9 | IC50 | 2 | — | |
SVDPMUQDJQIHAL
|
8.9 | IC50 | 2 | — | |
UUKGDBLVFLHJLM
|
8.9 | IC50 | 2 | — | |
XHHRGYCOEVNAKV
|
8.9 | Ki | 6 | Yes | |
ZLHFILGSQDJULK
|
8.9 | IC50 | 37 | Yes | |
GYOJAUPBIHPKFM
|
8.9 | IC50 | 2 | — | |
INWAPLGMARPPCH
|
8.9 | IC50 | 3 | — | |
LSOZVYDETZGJRK
|
8.9 | IC50 | 3 | — | |
NERGHRXOVVUXNP
|
8.9 | IC50 | 2 | — | |
XAQZJRAEQPCWMI
|
8.9 | IC50 | 3 | Yes | |
DTHIPVGUOHBTJC
|
8.8 | IC50 | 2 | — | |
GSWYQMZWPSIFDH
|
8.8 | IC50 | 3 | — | |
HLGQFYSTVZBBCM
|
8.8 | IC50 | 3 | — | |
OIDHYGPWCABWGM
|
8.8 | IC50 | 3 | — | |
RDMDYYYJDXIUDF
|
8.8 | IC50 | 2 | — | |
WFJYZRKNRWYRTN
|
8.8 | IC50 | 3 | — | |
XQWJBQQWWOWGQH
|
8.8 | IC50 | 2 | — | |
AWJSEDIXXHFUSS
|
8.8 | IC50 | 3 | — | |
GJSXBANTJATBDM
|
8.8 | IC50 | 2 | — | |
MBKBRIBQHFBRHO
|
8.8 | IC50 | 3 | — | |
MDHHYPFBVYJHPN
|
8.8 | IC50 | 6 | Yes | |
GCIKSSRWRFVXBI
|
8.8 | IC50 | 109 | Yes | |
FUIHJVJXGTVUJU
|
8.8 | IC50 | 3 | Yes | |
IKLMCSQBFDOMDW
|
8.8 | IC50 | 3 | — | |
KMFBAJNOTSSVEC
|
8.8 | IC50 | 2 | — | |
LCQYMDMUCJFFKN
|
8.8 | IC50 | 5 | Yes | |
LMBOMGUIBWYBDA
|
8.8 | IC50 | 3 | — | |
MVJMMLFMPWITEJ
|
8.8 | Ki | 110 | — | |
RKQAHDJYVWGPCS
|
8.8 | IC50 | 2 | — | |
VCFDMLBPASGZTP
|
8.8 | Ki | 38 | — | |
YKEMJPHTBLZSFI
|
8.8 | IC50 | 3 | — | |
VSUHZFYKALKPLP
|
8.8 | IC50 | 2 | — | |
ANTUVUVMQSIJBS
|
8.8 | IC50 | 3 | Yes | |
FTLGJGCPUAMLIH
|
8.8 | IC50 | 2 | — | |
NVWZWRFWZNYFRS
|
8.8 | IC50 | 2 | — | |
GABKCBKPNYHAJC
|
8.7 | IC50 | 3 | — | |
HEMLBLLRLPNMEZ
|
8.7 | IC50 | 2 | — | |
MNGNUDIQTBWWNA
|
8.7 | IC50 | 3 | — | |
PLSBOWQASGBKLJ
|
8.7 | IC50 | 2 | — | |
PQSAXJVMRVYGLM
|
8.7 | IC50 | 3 | — | |
QSWPJTLRYDNNBP
|
8.7 | IC50 | 3 | — | |
XGXROOYTEGFACC
|
8.7 | IC50 | 3 | — | |
NXUFRHVUTNXZQT
|
8.7 | IC50 | 2 | — | |
AJJYRLVECZPGED
|
8.7 | IC50 | 3 | — | |
IMDKLXHGHQNHPQ
|
8.7 | IC50 | 2 | — |