Target Details
| UniProt AC | O14965 |
|---|---|
| Gene Symbol | AURKA |
| Protein Name | Aurora kinase A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,119
- Clinical molecules 389
- Avg pChEMBL 7.5
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (2,119)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GTGQIIVTDZEGPK
|
9.1 | IC50 | 3 | — | |
HEBODLJXGULWNN
|
9.1 | IC50 | 3 | — | |
JMHMGIHHTONCMK
|
9.1 | IC50 | 3 | — | |
JXYHLSHMUKGXOI
|
9.1 | IC50 | 2 | — | |
PAPOXMYYOLMACK
|
9.1 | IC50 | 2 | — | |
SXRUTBTWKQVBSM
|
9.1 | IC50 | 3 | — | |
ZBLXMVSBOPAZEE
|
9.1 | IC50 | 2 | — | |
IDKYOQDTCCUVIN
|
9.1 | IC50 | 3 | — | |
OLDWHOFNZYPPSR
|
9.1 | IC50 | 2 | — | |
BXONPPLBOJAICG
|
9.1 | IC50 | 3 | — | |
KFKCUGPWEAJREP
|
9.1 | IC50 | 2 | — | |
TYTPWTMXQPOHQI
|
9.1 | IC50 | 2 | — | |
HOGWQTOSZMFOAJ
|
9.0 | IC50 | 2 | — | |
PXVPCLNOMYTQQA
|
9.0 | IC50 | 2 | — | |
UUVFRMLWZBOAOM
|
9.0 | IC50 | 3 | — | |
IILGZBCIXYOQFH
|
9.0 | IC50 | 2 | — | |
JPXOUJDDCUAQFV
|
9.0 | IC50 | 2 | — | |
LOGBBCVHUWZQRE
|
9.0 | IC50 | 2 | — | |
WVHAMWAJDWCCNB
|
9.0 | IC50 | 2 | — | |
BGCQKRIZWQNGJK
|
9.0 | IC50 | 2 | — | |
RKSDWJBFBPKMFN
|
9.0 | IC50 | 3 | — | |
SICPNVSSMIOAEC
|
9.0 | IC50 | 3 | — | |
ATUGFOWGVANOHQ
|
9.0 | Ki | 4 | Yes | |
BMYPGRZADREWCU
|
9.0 | IC50 | 3 | — | |
BRXHKUKMMZTVRE
|
9.0 | IC50 | 3 | — | |
FKBXSMMSZMPOPT
|
9.0 | IC50 | 2 | — | |
GUKNWLMFOBWSRH
|
9.0 | IC50 | 2 | Yes | |
HBBXYFBAAFTMQH
|
9.0 | IC50 | 2 | — | |
HELPFLHLGBGMOS
|
9.0 | Ki | 2 | — | |
IBBZLXWCFCMCKF
|
9.0 | IC50 | 3 | — | |
IBQHDBZMXPNKAU
|
9.0 | IC50 | 2 | Yes | |
JKUFJTIKVQADGJ
|
9.0 | IC50 | 2 | — | |
MVQSZXIVEQECJQ
|
9.0 | IC50 | 2 | — | |
OTACRQCAOBRLAZ
|
9.0 | Ki | 8 | Yes | |
OVSOFMFOYROLMC
|
9.0 | IC50 | 2 | — | |
PDULEZONFAQVLI
|
9.0 | IC50 | 3 | — | |
QQCDNHWVJDMTCC
|
9.0 | IC50 | 2 | — | |
SKQGEQYAZXPKCB
|
9.0 | IC50 | 3 | — | |
ULDURKNHYFYKMS
|
9.0 | IC50 | 3 | — | |
VFSDCFPRAHKMGQ
|
9.0 | IC50 | 2 | — | |
WJMWJDYFXSDIDZ
|
9.0 | IC50 | 2 | — | |
YQQZZYYQTCPEAS
|
9.0 | IC50 | 2 | — | |
AXENBBKNBUDYQA
|
9.0 | IC50 | 3 | — | |
BDDMFFMPRZTZGH
|
9.0 | IC50 | 2 | — | |
BXOCOVVDMXWPQN
|
9.0 | IC50 | 3 | — | |
FWCNPQPYGXFFSI
|
9.0 | IC50 | 3 | — | |
IVOSBLQIUULOJZ
|
9.0 | IC50 | 2 | — | |
LIQIOFRVUQMLKU
|
9.0 | IC50 | 2 | — | |
MYNMWFXSBRRDCA
|
9.0 | IC50 | 3 | — | |
RGLSQZGEAOHRTM
|
9.0 | IC50 | 3 | — |