Target Details
| UniProt AC | O14965 |
|---|---|
| Gene Symbol | AURKA |
| Protein Name | Aurora kinase A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,119
- Clinical molecules 389
- Avg pChEMBL 7.5
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (2,119)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XTDBGBVPMKZZHK
|
9.2 | IC50 | 2 | Yes | |
AADMVMUUAFAHRV
|
9.2 | IC50 | 2 | — | |
GXSLNZRYHCTIMQ
|
9.2 | IC50 | 2 | — | |
IGFVLPPIRBECDD
|
9.2 | IC50 | 2 | — | |
POQNJRCZSQACTE
|
9.2 | IC50 | 2 | — | |
QXNNCHKUKMPZRH
|
9.2 | IC50 | 2 | — | |
WYACPHRPKYXVTD
|
9.2 | IC50 | 2 | — | |
NZVDDFRUBIEKLV
|
9.2 | Ki | 20 | — | |
SFVVRJCZCCKAKZ
|
9.2 | IC50 | 2 | — | |
VPHVDXANMJOXMQ
|
9.2 | IC50 | 3 | — | |
XAGUVCIPGYLDFN
|
9.2 | IC50 | 2 | — | |
IWBOFXHEGIMYAM
|
9.2 | IC50 | 3 | — | |
IXXXRLXHQHLRSJ
|
9.2 | IC50 | 3 | — | |
KYEHLWMHQXZVMF
|
9.2 | IC50 | 2 | — | |
PGGKNOUMRNIDKJ
|
9.2 | IC50 | 2 | — | |
WNQHVGYFQUHRNW
|
9.2 | Ki | 4 | — | |
CITUHDBZOGJAEN
|
9.2 | IC50 | 3 | — | |
CWBIOTBDHJUHCV
|
9.2 | IC50 | 3 | — | |
UOYJLMIJVTUQOD
|
9.2 | IC50 | 2 | — | |
IUEUJHZZCUYXKU
|
9.2 | IC50 | 2 | — | |
GZBZDQBLAIACNB
|
9.2 | IC50 | 3 | — | |
LCHBJUVGCMYUMC
|
9.2 | IC50 | 2 | — | |
QCETXMLIFLYKQH
|
9.2 | IC50 | 3 | — | |
SLYMRFHIVVKAEL
|
9.2 | IC50 | 2 | — | |
BQOUQYBZXHHCIK
|
9.2 | IC50 | 2 | — | |
FFBJZTQMALZDTE
|
9.2 | IC50 | 2 | — | |
KGJQVQSYWYQQOD
|
9.2 | IC50 | 2 | — | |
JWYNPNNKXPDNQR
|
9.1 | IC50 | 2 | — | |
MZNBFJHMZMXTSD
|
9.1 | IC50 | 3 | — | |
QZHICJQAPASSMT
|
9.1 | IC50 | 2 | — | |
SWEZOINTKPVMEG
|
9.1 | IC50 | 3 | — | |
YWZXPHGLOMUDHA
|
9.1 | IC50 | 2 | — | |
HZCSYARAUKXOFF
|
9.1 | IC50 | 2 | — | |
BGKAQJOYFISGLZ
|
9.1 | IC50 | 2 | — | |
FMSSVKVRLRCICW
|
9.1 | IC50 | 2 | — | |
HAWOAWLBNXPWTR
|
9.1 | IC50 | 2 | — | |
LMGGXHWFXQXVKE
|
9.1 | IC50 | 2 | — | |
PJYYVACVVUDTRN
|
9.1 | IC50 | 3 | — | |
RNIRTUIZMXHJGS
|
9.1 | IC50 | 2 | — | |
RNIRTUIZMXHJGS
|
9.1 | IC50 | 3 | — | |
BLFRZPJRKJLHGU
|
9.1 | IC50 | 3 | — | |
GBLWEKVVBOPDQK
|
9.1 | IC50 | 2 | — | |
NMKNRNXEPYFWSY
|
9.1 | IC50 | 3 | — | |
RYYNGWLOYLRZLK
|
9.1 | IC50 | 45 | — | |
RHIXHHWKASAAHP
|
9.1 | IC50 | 2 | — | |
WPDWJWPDAWEUDW
|
9.1 | IC50 | 3 | — | |
XZTYFGBEDWNFPM
|
9.1 | IC50 | 3 | — | |
DCRRXSUQGXVDLQ
|
9.1 | IC50 | 2 | — | |
XWKILAVPLLWQTA
|
9.1 | IC50 | 2 | — | |
YOGFDHJWPOMSHT
|
9.1 | IC50 | 2 | — |