Target Details
| UniProt AC | O14965 |
|---|---|
| Gene Symbol | AURKA |
| Protein Name | Aurora kinase A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,119
- Clinical molecules 389
- Avg pChEMBL 7.5
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (2,119)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PLAVWQHGBMTMFR
|
9.4 | IC50 | 2 | — | |
PNSDQTZGJZEYEU
|
9.4 | IC50 | 2 | — | |
VNQGYSYYWYWSPN
|
9.4 | IC50 | 2 | — | |
WOHBHEXSHHPQIV
|
9.4 | Ki | 8 | Yes | |
XZEFTYTUTILRTG
|
9.4 | IC50 | 3 | — | |
OEFRWUPQSHQOMD
|
9.4 | IC50 | 2 | — | |
DHNFKQPWVFBZIL
|
9.4 | IC50 | 3 | — | |
IHDFFGIONOKCLR
|
9.4 | IC50 | 3 | — | |
NNDFRIHFDHSKHD
|
9.4 | IC50 | 3 | — | |
DQPVIVGCZVQZDO
|
9.4 | IC50 | 3 | — | |
VATUQWRZIIQRGK
|
9.4 | IC50 | 2 | — | |
FIZSPRJMYGKSMB
|
9.4 | IC50 | 2 | — | |
SHHVFBHRTMUGBM
|
9.4 | IC50 | 3 | — | |
RPMDNLSTGYONBC
|
9.3 | IC50 | 3 | — | |
COMSYOFZTVGRRK
|
9.3 | IC50 | 2 | — | |
JZIOOTOUNCFCCO
|
9.3 | IC50 | 2 | — | |
MMJLTRRVKQFACD
|
9.3 | IC50 | 2 | — | |
FVCBPYDMVVHXSV
|
9.3 | IC50 | 2 | — | |
OZKLXNJWZUXQAC
|
9.3 | IC50 | 3 | — | |
USUYXDKUCNQBKM
|
9.3 | IC50 | 3 | — | |
FYVFJSKWDZJJKR
|
9.3 | IC50 | 2 | — | |
JWLUINJKUPWLHG
|
9.3 | IC50 | 2 | — | |
LCTWFROMTHUGEH
|
9.3 | IC50 | 2 | — | |
VCASZZUAVHWYHQ
|
9.3 | IC50 | 3 | — | |
ZWRIWNSRFLBBOD
|
9.3 | IC50 | 3 | — | |
BYWLEEWVFXOXAG
|
9.3 | IC50 | 2 | — | |
GIBXNJNDDSOAHX
|
9.3 | IC50 | 2 | — | |
DDSBMKNXVLTBPK
|
9.3 | IC50 | 3 | — | |
FKRLYOFLOQRBNO
|
9.3 | IC50 | 2 | — | |
GRBADRHZGYZJTH
|
9.3 | IC50 | 3 | — | |
SZUFVMKRAKNXNR
|
9.3 | IC50 | 2 | — | |
WDDYOKLMIHMUSU
|
9.3 | IC50 | 2 | — | |
NFSWZORPOVHHLM
|
9.3 | IC50 | 2 | — | |
NXTQOFQOBODYSP
|
9.3 | IC50 | 2 | — | |
XUGCPDXHIQDAKV
|
9.3 | IC50 | 2 | — | |
ZLXRCPDTORAWNV
|
9.3 | IC50 | 2 | — | |
OIHRDLGLZDFHAD
|
9.2 | IC50 | 2 | — | |
SPCDTNUNXCPQPQ
|
9.2 | IC50 | 2 | — | |
KRUKDVBCEQTOCL
|
9.2 | IC50 | 3 | — | |
QOYWSCMDSDPETI
|
9.2 | IC50 | 2 | — | |
SNBMLCRFYZAAAX
|
9.2 | IC50 | 3 | — | |
SWYUPOALZWKXQY
|
9.2 | IC50 | 2 | — | |
YRQSEFHVBKRZFV
|
9.2 | IC50 | 2 | — | |
GEQPKDUYCDTQRY
|
9.2 | IC50 | 2 | — | |
JODNFBDDCMSPPR
|
9.2 | IC50 | 2 | — | |
VUEJUOUQJKHUSF
|
9.2 | IC50 | 2 | — | |
DWOLUZVOAOPIIX
|
9.2 | IC50 | 2 | — | |
IYDPFVSCKFTRQD
|
9.2 | IC50 | 2 | — | |
ORGQNRJTEJDZTI
|
9.2 | IC50 | 2 | — | |
SRNFZCPMRRFGPA
|
9.2 | IC50 | 2 | — |