Target Details
| UniProt AC | O14965 |
|---|---|
| Gene Symbol | AURKA |
| Protein Name | Aurora kinase A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,119
- Clinical molecules 389
- Avg pChEMBL 7.5
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (2,119)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RBVRSMCCUMHQRB
|
9.6 | IC50 | 2 | — | |
YAEXRFPBDXLXMG
|
9.6 | IC50 | 3 | — | |
BBNMVNJADAIHAK
|
9.6 | IC50 | 2 | — | |
CNFJGGPOIJUVKL
|
9.6 | IC50 | 2 | — | |
ABXUNSYTKULRPM
|
9.6 | IC50 | 2 | — | |
DHEDUDJQNPBXHX
|
9.6 | IC50 | 2 | — | |
RWBMPHFTXFAKIZ
|
9.6 | IC50 | 2 | — | |
WACBDIUIBDYGCE
|
9.6 | IC50 | 3 | — | |
AKYGBXZKHJOPDB
|
9.6 | IC50 | 3 | — | |
RXAZPQCDGXHCAO
|
9.6 | IC50 | 2 | — | |
KWBXLLQBOZJIAV
|
9.6 | IC50 | 2 | — | |
VWYGEDAFWDXUMQ
|
9.6 | IC50 | 3 | — | |
JWSHIVZYYNSBPC
|
9.5 | IC50 | 3 | — | |
JYUQCOURFHGOMR
|
9.5 | IC50 | 2 | — | |
VSIZGIFPGSTFOV
|
9.5 | IC50 | 3 | — | |
GPYJJUQMUZUDRC
|
9.5 | IC50 | 2 | — | |
HYBDRLATORKZNI
|
9.5 | IC50 | 3 | — | |
JMHMGIHHTONCMK
|
9.5 | IC50 | 2 | — | |
VVSYBPIXJIERDK
|
9.5 | IC50 | 2 | — | |
XISIJMIPHPQCQQ
|
9.5 | IC50 | 9 | — | |
KPFKWRJCTOGYCX
|
9.5 | IC50 | 2 | — | |
KXEUNUNXKXUREW
|
9.5 | IC50 | 2 | — | |
XQHCUHBVDXWRKR
|
9.5 | IC50 | 2 | — | |
YGEQQFLMLXRDQK
|
9.5 | IC50 | 3 | — | |
BTWIQOVBQBEGSN
|
9.5 | IC50 | 2 | — | |
ORMLOSONIQIDBI
|
9.5 | IC50 | 3 | — | |
LEKLEQSVVRJEHN
|
9.5 | IC50 | 2 | — | |
POBKWGYBFDTZBY
|
9.5 | IC50 | 2 | — | |
QSWPJTLRYDNNBP
|
9.5 | IC50 | 2 | — | |
GYEINYAKLFRDRF
|
9.5 | IC50 | 2 | — | |
SKTCDUXPKLCJIP
|
9.5 | IC50 | 3 | — | |
HAKWYGIXPYBWTK
|
9.5 | IC50 | 2 | — | |
RKZPJUYYKFXMLU
|
9.5 | IC50 | 3 | — | |
UZEGEPCLJOWZGN
|
9.4 | IC50 | 2 | — | |
CEONSWRDFKMFNM
|
9.4 | IC50 | 2 | — | |
MTPDPEHTPPGPLH
|
9.4 | IC50 | 3 | — | |
NQOIWUCLZREOSK
|
9.4 | IC50 | 2 | — | |
PUFIZMIVJDQOHA
|
9.4 | IC50 | 3 | — | |
RQYTYYKPVBSSQC
|
9.4 | IC50 | 2 | — | |
CVCLGNCOASWGPB
|
9.4 | IC50 | 2 | — | |
NWDPAGBWBJBPGW
|
9.4 | IC50 | 2 | — | |
YOZQOXRJRWBJBE
|
9.4 | IC50 | 2 | — | |
CXSMTMCUUMPVML
|
9.4 | IC50 | 2 | — | |
LLROFEFDEFKWQN
|
9.4 | IC50 | 3 | — | |
PWWRGGQDPGYVDM
|
9.4 | IC50 | 3 | — | |
FAEQSQDLHPQOMI
|
9.4 | IC50 | 2 | — | |
FFJNCCISXWZBSC
|
9.4 | IC50 | 2 | — | |
JEDGRRQUCXCFEZ
|
9.4 | IC50 | 3 | — | |
JQTUGUXQKTXVPW
|
9.4 | IC50 | 2 | — | |
NKKNQMFHKZEGQU
|
9.4 | IC50 | 5 | — |