Target Details
| UniProt AC | O14965 |
|---|---|
| Gene Symbol | AURKA |
| Protein Name | Aurora kinase A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,119
- Clinical molecules 389
- Avg pChEMBL 7.5
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (2,119)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LFVVQRUJKSZURN
|
9.8 | IC50 | 3 | — | |
MPLYXIRRQBHUMZ
|
9.8 | IC50 | 2 | — | |
XWICEOXKSZMQJY
|
9.8 | IC50 | 2 | — | |
DHNWCWGJFSTRBB
|
9.8 | IC50 | 3 | — | |
IABSWKZENVKESR
|
9.8 | IC50 | 3 | — | |
NRBGHJOLFXFDFP
|
9.8 | IC50 | 3 | — | |
RNGULOLZVZHPCT
|
9.8 | IC50 | 2 | — | |
SHTJDUVIHHPLRU
|
9.8 | IC50 | 2 | — | |
ARLBCCDWOPSKDJ
|
9.8 | IC50 | 3 | — | |
BZNBRLIMNHJECW
|
9.8 | IC50 | 2 | — | |
PSYMLFSTUXAGFZ
|
9.8 | IC50 | 3 | — | |
RHWHWWRJINHZQN
|
9.8 | IC50 | 2 | — | |
RWDHVFTXNBLJFJ
|
9.8 | IC50 | 2 | — | |
UFVBHPSYTMXORI
|
9.8 | IC50 | 2 | — | |
DLYWLUNYSQBOLW
|
9.7 | IC50 | 2 | — | |
JPDOHTKDIUCCPD
|
9.7 | IC50 | 2 | — | |
LBMOKRBEBYSURI
|
9.7 | IC50 | 3 | — | |
ODIUNKSOMOLOOF
|
9.7 | IC50 | 3 | — | |
PRQRZQNKZIWBFE
|
9.7 | IC50 | 2 | — | |
QJGKIKAFWQXPCF
|
9.7 | IC50 | 2 | — | |
RQMCICOFYAOUFP
|
9.7 | IC50 | 2 | — | |
SPWUNHDCOAYNOQ
|
9.7 | IC50 | 2 | — | |
VQTZMSIOEYJERT
|
9.7 | IC50 | 2 | — | |
ZKQGSMFEXARYCS
|
9.7 | IC50 | 3 | — | |
GBKAFRSEJQCGNT
|
9.7 | IC50 | 2 | — | |
GPPDWFNQVHJOEU
|
9.7 | IC50 | 3 | — | |
OSVOVHIYXDNBJQ
|
9.7 | IC50 | 3 | — | |
PJXUDKNHESNHGD
|
9.7 | IC50 | 2 | — | |
YXUPBHOIGGKRNR
|
9.7 | IC50 | 2 | — | |
ZYCYNVIAJAEECH
|
9.7 | IC50 | 2 | — | |
AJBCWROWNACASN
|
9.7 | IC50 | 3 | — | |
AJBCWROWNACASN
|
9.7 | IC50 | 3 | — | |
GTTSANJRVQIGFM
|
9.7 | IC50 | 3 | — | |
JGTLCWBXBNQZGX
|
9.7 | IC50 | 3 | — | |
JXOFZRFVAKUHDR
|
9.7 | IC50 | 2 | — | |
NLGYPTWGAPKFAZ
|
9.7 | IC50 | 3 | — | |
IHDFFGIONOKCLR
|
9.7 | IC50 | 3 | — | |
RFRCSMPUQCLUQP
|
9.7 | IC50 | 2 | — | |
ZTCGLAMYEAGAAN
|
9.7 | IC50 | 2 | — | |
FTMVCBNREGWDGS
|
9.7 | IC50 | 2 | — | |
HTRVDWTYRAEJCW
|
9.7 | IC50 | 3 | — | |
LAQKCNTWJTZLBG
|
9.7 | IC50 | 2 | — | |
LHDWVUBCEIVHFK
|
9.7 | IC50 | 2 | — | |
NXUJCUODKLXIPE
|
9.7 | IC50 | 2 | — | |
ODLVSMKOGBYEPO
|
9.7 | IC50 | 2 | — | |
QUXMKGGVROUWSP
|
9.7 | IC50 | 3 | — | |
UQDBHQAEMZNPSQ
|
9.7 | IC50 | 3 | — | |
ZLLVDXDXVWPFPN
|
9.7 | IC50 | 2 | — | |
FWHSZSDGPFVMOC
|
9.6 | IC50 | 3 | — | |
QJMIUPZFDRLJHJ
|
9.6 | IC50 | 2 | — |