Target Details
| UniProt AC | O14965 |
|---|---|
| Gene Symbol | AURKA |
| Protein Name | Aurora kinase A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,119
- Clinical molecules 389
- Avg pChEMBL 7.5
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (2,119)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HZUXHEBYLGLOGZ
|
8.0 | IC50 | 2 | — | |
AKIIIZOJWRPEPQ
|
8.0 | IC50 | 5 | Yes | |
BUKMSYYNNHEANR
|
8.0 | IC50 | 2 | — | |
CLOQRRBPZHLSQE
|
8.0 | IC50 | 3 | Yes | |
CNTCGRJDUJEUDG
|
8.0 | Ki | 37 | — | |
DBXGGXLBTWZXBB
|
8.0 | Ki | 39 | — | |
GBMDFZRFAMTRLI
|
8.0 | IC50 | 2 | — | |
HIJNIPAQZUMXON
|
8.0 | IC50 | 2 | — | |
HIXRSEFUZBICPP
|
8.0 | Kd | 2 | — | |
HMLDXQBTXVPSOC
|
8.0 | IC50 | 3 | — | |
KMWZKNHCFZNBFL
|
8.0 | Ki | 3 | Yes | |
LSEOXFVSQOHSDK
|
8.0 | Kd | 3 | — | |
MHCPAORAYMTGCZ
|
8.0 | Ki | 37 | — | |
NNQPYKAOGXIZBP
|
8.0 | IC50 | 2 | — | |
OPVKJVDDNDEKSB
|
8.0 | Kd | 2 | — | |
QRDRCIWCMVIMHC
|
8.0 | IC50 | 3 | — | |
RYROLHUONOCJPP
|
8.0 | IC50 | 2 | — | |
SBJRRILZYCCWJE
|
8.0 | IC50 | 5 | — | |
SRUYMJRFVGLQDV
|
8.0 | Ki | 37 | — | |
XKZINYYXWJEYEL
|
8.0 | Ki | 37 | — | |
HLXBUKYOKGQEDD
|
8.0 | Kd | 2 | — | |
XLUIYTJCFLMYKF
|
8.0 | IC50 | 2 | — | |
BCSHETJKMWOYNN
|
8.0 | IC50 | 2 | — | |
FGLDVWQEBUVALV
|
8.0 | IC50 | 3 | — | |
GCHPTPVYEQUDIU
|
8.0 | IC50 | 2 | — | |
GLDSKRNGVVYJAB
|
8.0 | IC50 | 16 | — | |
JZAIDLUIAGRFMY
|
8.0 | IC50 | 2 | — | |
MPCQRPKDRXWSSR
|
8.0 | Ki | 4 | Yes | |
NYZJWCNLQGNIQE
|
8.0 | IC50 | 2 | — | |
OAOPWYXDCLIWEH
|
8.0 | Kd | 2 | — | |
OSOQQRUVRRWBMV
|
8.0 | IC50 | 3 | — | |
QIKJAWWGNVSEHB
|
8.0 | IC50 | 2 | — | |
QQJKCGXOHWHBQV
|
8.0 | IC50 | 4 | — | |
QURBHJPQZDAPGP
|
8.0 | IC50 | 3 | — | |
RPSFIQJOUUTWRS
|
8.0 | IC50 | 3 | Yes | |
SGZZQKMOFHIDKW
|
8.0 | IC50 | 13 | — | |
SSERHUGYONZSKK
|
8.0 | IC50 | 2 | — | |
STTWKDVRVDYNAH
|
8.0 | Kd | 2 | — | |
VPEYPVPNDMIFEL
|
8.0 | IC50 | 3 | — | |
VWQOMDPIYKNCFJ
|
8.0 | IC50 | 3 | Yes | |
WHLKRBBRZJQSQQ
|
8.0 | IC50 | 2 | — | |
YHTMTLWBCNPEPE
|
8.0 | IC50 | 4 | — | |
HBJUFAHIACMPFY
|
8.0 | IC50 | 4 | — | |
GLSXPVFPHBFULR
|
7.9 | IC50 | 2 | — | |
MMVLETOTGHDVPQ
|
7.9 | IC50 | 7 | — | |
DIZTWKKXOXSRQF
|
7.9 | Kd | 2 | — | |
ABRVQCRUWGRURK
|
7.9 | IC50 | 2 | — | |
BQRYSUAKKHQWCB
|
7.9 | IC50 | 2 | — | |
CERFFPJDBQMQTN
|
7.9 | IC50 | 2 | — | |
HNXLEVKZEPXIAQ
|
7.9 | IC50 | 2 | — |