Target Details
| UniProt AC | O14965 |
|---|---|
| Gene Symbol | AURKA |
| Protein Name | Aurora kinase A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,119
- Clinical molecules 389
- Avg pChEMBL 7.5
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (2,119)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OMRUWHFZQGLMRI
|
8.1 | IC50 | 2 | — | |
ADDQRQHBRAHARB
|
8.1 | Ki | 2 | — | |
CAZDZVMSMCBBSO
|
8.1 | IC50 | 3 | — | |
CPFWYOIIPHITHV
|
8.1 | IC50 | 2 | — | |
FZVCMCRNWSWUCG
|
8.1 | Kd | 3 | — | |
GNSDDKAAHUFOKJ
|
8.1 | IC50 | 3 | — | |
GRXDRZBYCBQOFV
|
8.1 | Kd | 2 | — | |
GXJSLIOOPZRPEV
|
8.1 | Ki | 34 | — | |
JBYKCUNHSBWUPW
|
8.1 | IC50 | 2 | — | |
JYVCLVPNSVUQHC
|
8.1 | Kd | 2 | — | |
MXYMWTPPSBKBGN
|
8.1 | Kd | 2 | — | |
NFKMFNBKEOQNPZ
|
8.1 | Ki | 43 | — | |
NROKZPYRSOKBHT
|
8.1 | IC50 | 3 | Yes | |
NROKZPYRSOKBHT
|
8.1 | IC50 | 2 | — | |
OAJNZHZQLRZZSC
|
8.1 | IC50 | 3 | Yes | |
PDRMIURRJQICEV
|
8.1 | IC50 | 2 | — | |
QWJHWNIFEWOQTF
|
8.1 | IC50 | 5 | Yes | |
RBXYGQNZRVPDNB
|
8.1 | Ki | 34 | — | |
SUFQAOLKAMDVKJ
|
8.1 | IC50 | 3 | — | |
ISJYBLSITFIPEB
|
8.1 | IC50 | 3 | — | |
ZYJPIJHRIXUYCK
|
8.1 | IC50 | 2 | — | |
CVCJVUAHYHAMIA
|
8.1 | IC50 | 3 | — | |
WTPNSJYAYYXYNJ
|
8.1 | IC50 | 3 | — | |
XMRWQUJWAVDOIO
|
8.1 | IC50 | 2 | — | |
CDBRRCRVKIRWPN
|
8.1 | IC50 | 2 | — | |
FNFNFQPDKWQWMU
|
8.1 | IC50 | 2 | — | |
VBWCCTREXYTDOA
|
8.1 | IC50 | 2 | — | |
AOTUWXLVFBXKRO
|
8.1 | IC50 | 2 | — | |
OPVKJVDDNDEKSB
|
8.1 | Kd | 2 | — | |
PNFSXOCCWZKQET
|
8.1 | IC50 | 2 | — | |
AANVTLVNTUEXNM
|
8.1 | IC50 | 3 | Yes | |
BQLIAGXOCFHIGO
|
8.1 | IC50 | 3 | — | |
FAYAUAZLLLJJGH
|
8.1 | IC50 | 36 | Yes | |
HJKIGCOQVAUXEZ
|
8.1 | IC50 | 2 | — | |
KJVHTJKPBZOBPJ
|
8.1 | Ki | 4 | Yes | |
KLKOJHYRAITDCX
|
8.1 | IC50 | 2 | — | |
KZBSEJKXWKPCLO
|
8.1 | Kd | 3 | — | |
MHBFJQBMIDGZOZ
|
8.1 | IC50 | 2 | — | |
NVJBRKUSNQZNKX
|
8.1 | IC50 | 3 | Yes | |
NYMXQEKCEGCXNT
|
8.1 | IC50 | 3 | Yes | |
OJYFHTZIIPZQCE
|
8.1 | Kd | 2 | — | |
SJJYWHYLVWAUQL
|
8.1 | Ki | 2 | — | |
VAKWGLDYQAWDPS
|
8.1 | Ki | 3 | Yes | |
VCHQRSNNPYKZBM
|
8.1 | IC50 | 2 | — | |
XEUIIWAFFDHEEJ
|
8.1 | IC50 | 2 | — | |
XQNMCONHYXAHKS
|
8.1 | IC50 | 3 | — | |
YYFZPPMJHCVHFH
|
8.1 | Kd | 2 | — | |
ZUXFIRWLAQBCCS
|
8.1 | IC50 | 8 | Yes | |
CKSFNWDGZCXQON
|
8.0 | IC50 | 2 | — | |
MLWHQHRPLFMZHY
|
8.0 | IC50 | 2 | — |