Target Details
| UniProt AC | O14965 |
|---|---|
| Gene Symbol | AURKA |
| Protein Name | Aurora kinase A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,119
- Clinical molecules 389
- Avg pChEMBL 7.5
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (2,119)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZYURNHOEBWWJHI
|
8.2 | IC50 | 2 | Yes | |
AOLZRAWEDMEAQY
|
8.2 | IC50 | 2 | — | |
GAVSAOOAIYZEHU
|
8.2 | IC50 | 2 | — | |
UIAQHDUGAOFVJM
|
8.2 | IC50 | 2 | — | |
ULOLUGXMKLIZGE
|
8.2 | IC50 | 8 | Yes | |
VIVMIDXUVLTISY
|
8.2 | IC50 | 2 | — | |
ADLPKFFMGIJZIM
|
8.2 | Ki | 44 | — | |
AMMZKHYVESSTRS
|
8.2 | IC50 | 2 | — | |
MCCCQFAOMZMZKE
|
8.2 | Ki | 52 | — | |
NESRKEKGRKLXJB
|
8.2 | IC50 | 3 | — | |
OPVKJVDDNDEKSB
|
8.2 | Kd | 2 | — | |
QPORZABOFXPRHM
|
8.2 | Ki | 18 | — | |
ROIWTEBVYRJZEG
|
8.2 | Ki | 3 | — | |
ULHGAQSVFPOUDY
|
8.2 | Ki | 43 | — | |
UVNLAMSMBMXIJB
|
8.2 | Kd | 2 | — | |
XBYVOPRDASFDMY
|
8.2 | Ki | 42 | — | |
FNPQADNIXKBYIS
|
8.2 | Kd | 2 | — | |
JXCWQMODNUZVKT
|
8.2 | IC50 | 3 | — | |
KFYFFELQRLSBEN
|
8.2 | IC50 | 2 | — | |
HMUXYNLHZILXOH
|
8.2 | IC50 | 3 | — | |
LTTWDGKJGMQNHP
|
8.2 | IC50 | 3 | — | |
CNDJXGSDDHGEBJ
|
8.2 | IC50 | 2 | — | |
DAKDDXUSLPNQJJ
|
8.2 | IC50 | 2 | — | |
DQRVOAFQMMLWCP
|
8.2 | Kd | 3 | — | |
DVEOTEMULYJRLQ
|
8.2 | IC50 | 2 | — | |
GTWKARFQAYQPGO
|
8.2 | IC50 | 2 | — | |
HJVDQPRJANOXIX
|
8.2 | IC50 | 10 | — | |
MEKHYJNJENZTPN
|
8.2 | IC50 | 3 | Yes | |
MEKHYJNJENZTPN
|
8.2 | IC50 | 2 | — | |
MQWHYEKERKXFQY
|
8.2 | Kd | 2 | — | |
NKQFVOKSVRQZKX
|
8.2 | IC50 | 2 | — | |
PASPLONSFSXGKA
|
8.2 | IC50 | 2 | — | |
QZEWXOZPGITETL
|
8.2 | IC50 | 2 | — | |
SCMPDMAJYNSKMW
|
8.2 | Kd | 3 | — | |
VIDVOURISMXBLG
|
8.2 | IC50 | 3 | — | |
WPASUZBJIGBQSX
|
8.2 | IC50 | 2 | — | |
XQBLYDOGTIKRAE
|
8.2 | Kd | 2 | — | |
ZBPGILZGNLFHOC
|
8.2 | IC50 | 2 | — | |
FYWNMALNWQLLBJ
|
8.1 | IC50 | 2 | — | |
LOLPPWBBNUVNQZ
|
8.1 | IC50 | 97 | Yes | |
TYZWLLLNCLERKU
|
8.1 | IC50 | 3 | — | |
XGLWHPMFXKSELJ
|
8.1 | IC50 | 3 | — | |
GBJVVSCPOBPEIT
|
8.1 | IC50 | 13 | Yes | |
INIPMXIFCLHYIN
|
8.1 | IC50 | 2 | — | |
KOOZPNYTOCFUNJ
|
8.1 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
8.1 | IC50 | 408 | — | |
QJOLFMLQXIPTTF
|
8.1 | IC50 | 3 | — | |
VYOUAZSLWNSVRL
|
8.1 | IC50 | 3 | — | |
JYTYZRSXADUJAY
|
8.1 | IC50 | 2 | — | |
KDFQZJLGQYVRDD
|
8.1 | IC50 | 2 | — |