Target Details
| UniProt AC | O14965 |
|---|---|
| Gene Symbol | AURKA |
| Protein Name | Aurora kinase A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,119
- Clinical molecules 389
- Avg pChEMBL 7.5
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (2,119)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JKJUIAJEDWYGAG
|
8.3 | IC50 | 3 | — | |
MZKUHSLTLQVOKM
|
8.3 | Kd | 2 | — | |
NDJAPUTXCKBOMQ
|
8.3 | IC50 | 2 | — | |
NQFJXYKOQSRMCX
|
8.3 | Ki | 4 | Yes | |
NRTFVVVPFDOHFK
|
8.3 | IC50 | 2 | — | |
OWRXHGAFWZFFCW
|
8.3 | Ki | 113 | — | |
PASPLONSFSXGKA
|
8.3 | IC50 | 2 | — | |
RYAVJHIPOWNWDE
|
8.3 | Ki | 38 | — | |
SBCKWBIUBYZDRL
|
8.3 | IC50 | 2 | — | |
SPTNJNJCNRTHDY
|
8.3 | IC50 | 3 | Yes | |
UMIUXVPQKJLPJE
|
8.3 | Ki | 4 | — | |
UZWFLOSUVZITCB
|
8.3 | IC50 | 2 | Yes | |
VEJCMMPVTMQFME
|
8.3 | Ki | 8 | Yes | |
VKBFHTIUXUCYRQ
|
8.3 | Ki | 66 | — | |
XMSFPGDGANKHJW
|
8.3 | IC50 | 2 | — | |
YRNDLUNPBSSFMF
|
8.3 | IC50 | 3 | — | |
ZXAGZULZCKUUKQ
|
8.3 | IC50 | 2 | — | |
CJSJFNXXOCNUIQ
|
8.3 | Kd | 2 | — | |
HJQMKDZFPSWOEL
|
8.3 | IC50 | 2 | — | |
NHMACPMXYHTADL
|
8.3 | Ki | 3 | Yes | |
ZJTCESMUJZZNAL
|
8.3 | IC50 | 3 | — | |
LXAVLHJMLKIDME
|
8.3 | Ki | 3 | — | |
IBAUSYCHSXHDOA
|
8.3 | IC50 | 3 | — | |
YNNQCQWREXRBLV
|
8.3 | IC50 | 2 | — | |
LPSBYKLLJOVSHM
|
8.3 | IC50 | 2 | — | |
MXPLKNYFRWTHPW
|
8.3 | IC50 | 2 | — | |
QWDOEIJNIDENOC
|
8.3 | IC50 | 3 | — | |
WWOGYCVPNPHFGR
|
8.3 | IC50 | 2 | — | |
YISSDERVCVSJHT
|
8.3 | IC50 | 2 | — | |
HHFBDROWDBDFBR
|
8.2 | IC50 | 40 | Yes | |
SMOTZGTWZKCZAR
|
8.2 | Kd | 2 | — | |
SVGLHBXJLVCYTC
|
8.2 | IC50 | 2 | — | |
GXDMNAKMJVMWKQ
|
8.2 | IC50 | 5 | Yes | |
WTZPLLLUSQHZPS
|
8.2 | IC50 | 3 | — | |
FPKSFXFWECAIBR
|
8.2 | IC50 | 6 | Yes | |
KVMFMAFRXJBOKN
|
8.2 | IC50 | 2 | — | |
OPQNQTLSYVBRSX
|
8.2 | IC50 | 3 | — | |
QDKAHXFKNDNBHM
|
8.2 | IC50 | 2 | — | |
AKWLDQDWZNJYKL
|
8.2 | IC50 | 14 | — | |
BRXHKUKMMZTVRE
|
8.2 | IC50 | 3 | — | |
DEYRVWAAPWPOND
|
8.2 | IC50 | 3 | Yes | |
HCNZXJZRFQSKII
|
8.2 | IC50 | 2 | — | |
JNRTVZLIHFRYQO
|
8.2 | IC50 | 2 | Yes | |
KGHHVSJZWGWWDG
|
8.2 | IC50 | 4 | Yes | |
KTRJFPLINHVYDK
|
8.2 | Ki | 3 | Yes | |
KZDYTAXBOFTVGN
|
8.2 | IC50 | 3 | — | |
NKWGBOOLJXYPQR
|
8.2 | Ki | 2 | — | |
QZTBLEFQOCINTB
|
8.2 | IC50 | 3 | Yes | |
VKVBESYYODLWDZ
|
8.2 | IC50 | 2 | — | |
ZIZAJYWIUBTSRC
|
8.2 | Kd | 2 | — |