Target Details
| UniProt AC | O14965 |
|---|---|
| Gene Symbol | AURKA |
| Protein Name | Aurora kinase A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,119
- Clinical molecules 389
- Avg pChEMBL 7.5
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (2,119)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VNLDWMOEKZFKDP
|
8.4 | IC50 | 3 | — | |
BOWYXGHFMQMXPT
|
8.4 | Ki | 9 | — | |
CPGPEVNIOCXOPN
|
8.4 | IC50 | 3 | — | |
DQXCRLJTGIDAES
|
8.4 | IC50 | 2 | — | |
GHXCSPGXRVESNT
|
8.4 | IC50 | 2 | — | |
GZEGBHAXGLPTQY
|
8.4 | IC50 | 2 | — | |
IBWNGAFCNXNEDG
|
8.4 | Ki | 4 | Yes | |
KHDLZWDZNAKTKK
|
8.4 | Ki | 4 | Yes | |
KNOIFPSQNXJZDE
|
8.4 | IC50 | 3 | — | |
LDGFTLHOBZCPLF
|
8.4 | Ki | 2 | — | |
NRRLLJHNIQEBIO
|
8.4 | Kd | 2 | — | |
QHLGSHJIJSOCMR
|
8.4 | IC50 | 3 | — | |
QNOOVTZVMOOSAW
|
8.4 | IC50 | 4 | — | |
QNOOVTZVMOOSAW
|
8.4 | IC50 | 3 | — | |
ROGHHIGHHTZCFT
|
8.4 | IC50 | 3 | Yes | |
RYYNGWLOYLRZLK
|
8.4 | Ki | 104 | — | |
SYCRYYILCMOTOI
|
8.4 | IC50 | 3 | — | |
UYJNQQDJUOUFQJ
|
8.4 | IC50 | 68 | — | |
VAOPKWIEANDPSM
|
8.4 | Kd | 2 | — | |
VQBZFHKHISYRMO
|
8.4 | Ki | 2 | — | |
XDRKRJZKFZAPIW
|
8.4 | Kd | 2 | — | |
XDTMWNUVKUHOQV
|
8.4 | IC50 | 2 | — | |
XLSPYLMTRXPYKY
|
8.4 | IC50 | 13 | — | |
YBOBJBRACZBMOB
|
8.4 | IC50 | 2 | — | |
YTRICIMLLKPESG
|
8.4 | IC50 | 6 | — | |
YXEIECLOAMHVCH
|
8.4 | IC50 | 3 | Yes | |
ZCCJKVBTHCOISJ
|
8.4 | Ki | 46 | — | |
DABIENOBUSCARE
|
8.4 | Kd | 2 | — | |
ICODOOXDNPOINQ
|
8.4 | IC50 | 3 | — | |
MVVLRGOQAYKEMN
|
8.4 | IC50 | 2 | — | |
MVVLRGOQAYKEMN
|
8.4 | IC50 | 2 | — | |
GAAHSFKFIMENOG
|
8.4 | IC50 | 3 | Yes | |
MXHHONGZVDTFNW
|
8.4 | IC50 | 2 | — | |
QHLGSHJIJSOCMR
|
8.4 | IC50 | 2 | — | |
QXTIKAMWRHHMBU
|
8.4 | IC50 | 3 | — | |
UNRMMILBIIITEU
|
8.4 | IC50 | 3 | — | |
JRJLSKJAGSYHAP
|
8.3 | IC50 | 3 | — | |
SIDSSTAVUKNHFG
|
8.3 | Kd | 2 | — | |
KSFGFFQQMLCHJC
|
8.3 | IC50 | 3 | — | |
CRFHZXHUGPCWJA
|
8.3 | IC50 | 8 | — | |
MSISHOSYNKFLMZ
|
8.3 | IC50 | 3 | — | |
WGGOYMCUJRCWRJ
|
8.3 | IC50 | 3 | — | |
YFTUDCDZHZYZAB
|
8.3 | IC50 | 2 | — | |
BFSNADDVVFYGDC
|
8.3 | Kd | 2 | — | |
BKIGTXQKUBIVPY
|
8.3 | IC50 | 2 | — | |
BTZIOWUABPKONC
|
8.3 | IC50 | 2 | — | |
DRDUZQHVFDFHIY
|
8.3 | IC50 | 3 | Yes | |
FPDMCBWYLQMASE
|
8.3 | IC50 | 2 | — | |
GYZHPLHOIMYBJI
|
8.3 | Ki | 2 | — | |
IVUGFMLRJOCGAS
|
8.3 | IC50 | 9 | — |