Target Details
| UniProt AC | O14965 |
|---|---|
| Gene Symbol | AURKA |
| Protein Name | Aurora kinase A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,119
- Clinical molecules 389
- Avg pChEMBL 7.5
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (2,119)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NNQHKTWARZSGTQ
|
11.0 | Kd | 7 | — | |
QTTGVGLTCILDCA
|
11.0 | Kd | 7 | — | |
SRJJNRIRROSSLD
|
10.5 | IC50 | 2 | — | |
TUVCZMWCKOCSGF
|
10.5 | IC50 | 2 | — | |
HIUMPNPHWNCFBW
|
10.3 | IC50 | 3 | — | |
SZCJQZJURBSEEN
|
10.3 | IC50 | 2 | — | |
BNTYNTVACAGJNE
|
10.2 | IC50 | 2 | — | |
OVWZZXGBBZJATH
|
10.2 | IC50 | 3 | — | |
TUVCZMWCKOCSGF
|
10.2 | IC50 | 3 | — | |
LCVIRAZGMYMNNT
|
10.2 | IC50 | 4 | — | |
LCVIRAZGMYMNNT
|
10.2 | IC50 | 20 | — | |
GTUAZZUFAUMXII
|
10.2 | IC50 | 2 | — | |
RFRCSMPUQCLUQP
|
10.2 | IC50 | 2 | — | |
RHELVXGNWNTPJF
|
10.2 | IC50 | 3 | — | |
CFSJJIBVJMSQIL
|
10.1 | IC50 | 2 | — | |
LSBLRFKCBQDXLO
|
10.1 | IC50 | 2 | — | |
NHLHBOLWWGNMJH
|
10.1 | IC50 | 2 | — | |
RQAXQHGKLHCEHQ
|
10.1 | IC50 | 2 | — | |
SRJJNRIRROSSLD
|
10.1 | IC50 | 3 | — | |
VHSSUFWQNFHOQT
|
10.1 | IC50 | 3 | — | |
LDFNTCCSAZUOGI
|
10.1 | IC50 | 2 | — | |
OXHFPLUADZAODN
|
10.1 | IC50 | 2 | — | |
ROJRDYDJKQGLRH
|
10.1 | IC50 | 3 | — | |
TXCWDJYJHQBALS
|
10.1 | IC50 | 2 | — | |
GTUAZZUFAUMXII
|
10.0 | IC50 | 2 | — | |
RCBPCGVUXHCRAA
|
10.0 | IC50 | 2 | — | |
ASVHLUISRWYGFL
|
10.0 | IC50 | 3 | — | |
FURXQBPRWUDWOM
|
10.0 | IC50 | 2 | — | |
ITKXNAMPORNHCX
|
10.0 | IC50 | 2 | — | |
OVECHGPXFIKXEK
|
10.0 | IC50 | 3 | — | |
PELODSQJHQJMMD
|
10.0 | IC50 | 2 | — | |
RGXAJUCULIIOCG
|
10.0 | IC50 | 2 | — | |
XZHGTQKZIVZJHA
|
10.0 | IC50 | 2 | — | |
JMSLGFQQYRJYBH
|
9.9 | IC50 | 2 | — | |
KVVZDQBHKUCWQF
|
9.9 | IC50 | 3 | — | |
LJMKRAKDJVPMIO
|
9.9 | IC50 | 3 | — | |
MCVWAVHQVAZAKZ
|
9.9 | IC50 | 3 | — | |
NCPSMNWGGLQFPN
|
9.9 | IC50 | 2 | — | |
PZWGYFJPWNXLGT
|
9.9 | IC50 | 3 | — | |
RVKICAVHAJMKKD
|
9.9 | IC50 | 2 | — | |
VXJNQGXNBJPYRH
|
9.9 | IC50 | 2 | — | |
WOSUZOOSGPAWAC
|
9.9 | IC50 | 3 | — | |
WUTICGGSWNCYCY
|
9.9 | IC50 | 2 | — | |
YGQJBWJOHRVWHU
|
9.9 | IC50 | 3 | — | |
WACBDIUIBDYGCE
|
9.9 | IC50 | 3 | — | |
WOMKQOXPOGODKV
|
9.9 | IC50 | 3 | — | |
ZIAKJYHNHPITCS
|
9.9 | IC50 | 2 | — | |
FCZJOUALYCXWEB
|
9.8 | IC50 | 2 | — | |
IDGLADROFDGGQO
|
9.8 | IC50 | 2 | — | |
BMYPVSWCQCKWHI
|
9.8 | IC50 | 3 | — |