Target Details
| UniProt AC | O14929 |
|---|---|
| Gene Symbol | HAT1 |
| Protein Name | Histone acetyltransferase type B catalytic subunit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21183 (HAT1_C) PF10394 (Hat1_N) |
Summary
- Multi-target molecules 168
- Clinical molecules 0
- Avg pChEMBL 6.98
KEGG Pathways (2)
Active Molecules (168)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VUNIVHBJGHPCRI
|
7.3 | IC50 | 2 | — | |
FMIRMIPUPDECHV
|
7.3 | IC50 | 2 | — | |
PZMDZHITJJVGOE
|
7.3 | IC50 | 2 | — | |
KIRQWNADLAWJTG
|
7.2 | IC50 | 2 | — | |
BWEUTLKRALRPIQ
|
7.2 | IC50 | 2 | — | |
RIEJRXHPNFTDTB
|
7.2 | IC50 | 2 | — | |
BRDWGDCKTCQZHX
|
7.2 | IC50 | 2 | — | |
RBKUMEDNCTZKKV
|
7.2 | IC50 | 2 | — | |
ZAEXPXKGBRISBD
|
7.2 | IC50 | 2 | — | |
VJAWCSZJCQCSII
|
7.2 | IC50 | 2 | — | |
CYSITNKCPSLBOI
|
7.1 | IC50 | 2 | — | |
YZLHFVLRIDPTGT
|
7.1 | IC50 | 2 | — | |
WAMYZVOQTGAIAL
|
7.1 | IC50 | 2 | — | |
XGBNNEZVBIKAQY
|
7.1 | IC50 | 2 | — | |
ZXNRDVKXEACFMY
|
7.0 | IC50 | 2 | — | |
YZLHFVLRIDPTGT
|
7.0 | IC50 | 2 | — | |
MPTLMMCZHBKKSK
|
7.0 | IC50 | 2 | — | |
RYPHRIMKBWOBND
|
6.9 | IC50 | 2 | — | |
VEDJDLCMIXFLOX
|
6.9 | IC50 | 2 | — | |
LCZQNVZZLYLCLI
|
6.9 | IC50 | 2 | — | |
NJRFQVLIBLFGSD
|
6.9 | IC50 | 2 | — | |
AIGITZYSZNQTRP
|
6.9 | IC50 | 2 | — | |
PCYHEEQFXWHJDX
|
6.9 | IC50 | 2 | — | |
UMNKVLIESSDBJD
|
6.9 | IC50 | 2 | — | |
PAACZDGFYPGJSR
|
6.8 | IC50 | 2 | — | |
LRYNUODVDYSXHA
|
6.8 | IC50 | 2 | — | |
LRYNUODVDYSXHA
|
6.8 | IC50 | 2 | — | |
LANAKWBBQQVXFH
|
6.8 | IC50 | 2 | — | |
RIEJRXHPNFTDTB
|
6.8 | IC50 | 2 | — | |
HBOYJKDHPQOSOD
|
6.8 | IC50 | 2 | — | |
RBKUMEDNCTZKKV
|
6.7 | IC50 | 2 | — | |
ZCCPLJOKGAACRT
|
6.7 | Kd | 599 | — | |
CJBSZRRAPOGOGV
|
6.7 | IC50 | 2 | — | |
FLDRABMKVYNECQ
|
6.7 | IC50 | 2 | — | |
BQGXWMKUWPUXDO
|
6.7 | IC50 | 2 | — | |
RMKPSBLMNABFQY
|
6.7 | IC50 | 2 | — | |
BYFPXEICZVXFNB
|
6.7 | IC50 | 2 | — | |
LCXWSQLEGBEFSL
|
6.7 | IC50 | 2 | — | |
OJALLZBPDOMARU
|
6.7 | IC50 | 2 | — | |
DDNUAYKNTZWGNB
|
6.7 | IC50 | 2 | — | |
OJALLZBPDOMARU
|
6.6 | IC50 | 2 | — | |
PREKJLYPZPHGBS
|
6.6 | IC50 | 2 | — | |
VATKPQINTZGLTF
|
6.6 | IC50 | 2 | — | |
FRJIYEMWRIVSAU
|
6.6 | IC50 | 2 | — | |
RCCMPGJSLYZGCM
|
6.6 | IC50 | 2 | — | |
JHNYAHKUHMLTKC
|
6.5 | IC50 | 2 | — | |
SNNIHRFXLBXFQB
|
6.5 | IC50 | 2 | — | |
YTJSIMSRVUXEEW
|
6.5 | IC50 | 2 | — | |
ZEGFDPWUAOPASA
|
6.5 | IC50 | 2 | — | |
XGBNNEZVBIKAQY
|
6.5 | IC50 | 2 | — |