Target Details
| UniProt AC | O14920 |
|---|---|
| Gene Symbol | IKBKB |
| Protein Name | Inhibitor of nuclear factor kappa-B kinase subunit beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18397 (IKBKB_SDD) PF12179 (IKKbetaNEMObind) PF00069 (Pkinase) |
Summary
- Multi-target molecules 411
- Clinical molecules 17
- Avg pChEMBL 8.02
KEGG Pathways (60)
- Acute myeloid leukemia
- Adipocytokine signaling pathway
- Alcoholic liver disease
- Alzheimer disease
- Antifolate resistance
- Apoptosis
- B cell receptor signaling pathway
- C-type lectin receptor signaling pathway
- Cadherin signaling
- Chagas disease
- Chemical carcinogenesis - reactive oxygen species
- Chemokine signaling pathway
- Chronic myeloid leukemia
- Coronavirus disease - COVID-19
- Cytosolic DNA-sensing pathway
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- Fluid shear stress and atherosclerosis
- FoxO signaling pathway
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human T-cell leukemia virus 1 infection
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- IL-17 signaling pathway
- Influenza A
- Insulin resistance
- Insulin signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- MicroRNAs in cancer
- NF-kappa B signaling pathway
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Non-alcoholic fatty liver disease
- Osteoclast differentiation
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Prostate cancer
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Salmonella infection
- Shigellosis
- Small cell lung cancer
- T cell receptor signaling pathway
- TNF signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Type II diabetes mellitus
- Yersinia infection
- mTOR signaling pathway
Associated Diseases (1)
Active Molecules (411)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BKTQMCJLIKFGMJ
|
8.3 | Ki | 2 | — | |
ZOTMWAXVCBVWLO
|
8.3 | Ki | 2 | — | |
MXYAWDJBECRKLX
|
8.3 | IC50 | 6 | — | |
POVJWLXOAPPGME
|
8.3 | IC50 | 2 | — | |
SITLTVJDDVYTEN
|
8.3 | IC50 | 2 | — | |
GFLIQOFGXIPKRF
|
8.3 | Ki | 2 | — | |
YPPBYVJGQOGUSY
|
8.3 | Ki | 2 | — | |
CUWHKXADIYQZNO
|
8.2 | Ki | 2 | — | |
APRXYRORERCWAV
|
8.2 | IC50 | 2 | — | |
HBKASJKFEFLCPR
|
8.2 | IC50 | 2 | — | |
QBYYCHRRPPTEBG
|
8.2 | IC50 | 2 | — | |
IHJGLZRMTXXFEI
|
8.2 | Ki | 2 | — | |
ZPQGWIWZWZNROO
|
8.2 | IC50 | 6 | — | |
CCWWRYWEYAHFOL
|
8.2 | IC50 | 2 | — | |
IACXHGMTYKHWIP
|
8.2 | Ki | 2 | — | |
SSKFWKZRFZKTNE
|
8.2 | IC50 | 2 | — | |
WESZAXMBDDQWNG
|
8.2 | IC50 | 2 | — | |
DZDOYHVGPBMQIF
|
8.1 | IC50 | 5 | — | |
VSXRUMKXZQAYQC
|
8.1 | Ki | 2 | — | |
WIBJQYDYJUACSD
|
8.1 | IC50 | 7 | — | |
KRSGQERAJYCQMK
|
8.1 | Ki | 2 | — | |
YRIZQQKMLAOLSN
|
8.1 | Ki | 2 | — | |
PBEDKMOIZRXVCC
|
8.1 | Ki | 2 | — | |
GARGJFCAYIKMFS
|
8.1 | IC50 | 2 | — | |
HWADPPKZZYESMF
|
8.1 | IC50 | 2 | — | |
RDTKDSIRKDXUTE
|
8.1 | IC50 | 2 | — | |
VBFOQJUDSYRBDR
|
8.1 | IC50 | 2 | — | |
YFSYLICIZSSYBB
|
8.1 | IC50 | 2 | — | |
ZEVAYPOLTQWGHH
|
8.1 | IC50 | 2 | — | |
IFYDROJSRZHNOS
|
8.1 | IC50 | 7 | — | |
UDOPKESZEISBPX
|
8.1 | Ki | 2 | — | |
DYVFBWXIOCLHPP
|
8.1 | IC50 | 2 | — | |
ZAUQKMTUOLGTHT
|
8.1 | IC50 | 2 | — | |
APRXYRORERCWAV
|
8.1 | IC50 | 2 | — | |
ULTCRVJUAZCGPP
|
8.1 | IC50 | 5 | — | |
HYWKTDGSRPVHPB
|
8.0 | IC50 | 4 | — | |
CQCYWIZNPPGUKF
|
8.0 | Ki | 2 | — | |
OAJXWZOCHNZHSY
|
8.0 | Ki | 2 | — | |
BFXYIBREKSWTFK
|
8.0 | IC50 | 2 | — | |
KTPZTVBPMOHXFD
|
8.0 | Ki | 2 | — | |
LUAWBDVVBXMLEL
|
8.0 | IC50 | 7 | — | |
HDJJCDBHJXIVLV
|
8.0 | Ki | 2 | — | |
VTVFVCAHYRFAGQ
|
8.0 | Ki | 2 | — | |
BAAUCSNGBWGPNR
|
8.0 | Ki | 2 | — | |
JNXWYRLSXQVBBC
|
8.0 | IC50 | 2 | — | |
MDTKQKJDAXYFCW
|
8.0 | IC50 | 2 | — | |
SOFBJAGASYHSSD
|
8.0 | IC50 | 2 | — | |
WVAGWWGCPIPVSM
|
8.0 | IC50 | 2 | — | |
WUSLSBATAJISAC
|
8.0 | Ki | 2 | — | |
DJCIBWVKUOLMEK
|
7.9 | IC50 | 5 | — |