Target Details
| UniProt AC | O14757 |
|---|---|
| Gene Symbol | CHEK1 |
| Protein Name | Serine/threonine-protein kinase Chk1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 617
- Clinical molecules 26
- Avg pChEMBL 7.21
KEGG Pathways (6)
Associated Diseases (1)
Active Molecules (617)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YTGZRKKSIATJSK
|
6.8 | IC50 | 5 | — | |
FJQLYBZQSJEUED
|
6.8 | IC50 | 4 | — | |
WOSVQDVRYSIVTA
|
6.8 | IC50 | 2 | — | |
ZHIDPKVNWVGWNZ
|
6.8 | IC50 | 5 | — | |
MXVRLIJSNHJYSJ
|
6.7 | IC50 | 2 | — | |
RDRCDECEAGIASX
|
6.7 | IC50 | 2 | — | |
YROWXHNDJJAODS
|
6.7 | IC50 | 5 | — | |
FTFDOZLQPLTYBX
|
6.7 | IC50 | 7 | Yes | |
QPGSWTIJTZFCHL
|
6.7 | IC50 | 4 | — | |
CHZVKBHCILLIQS
|
6.7 | IC50 | 4 | — | |
HZASIAXCPXTISQ
|
6.7 | IC50 | 2 | — | |
UEFCSGDOOJJXTN
|
6.7 | IC50 | 46 | — | |
WKRLSDYBEGDEDI
|
6.7 | IC50 | 4 | — | |
CSQQBGXAZRAXLV
|
6.7 | Ki | 3 | — | |
FNLZQIHHIXKRNH
|
6.7 | IC50 | 2 | — | |
GHWMQXIAILGGTF
|
6.7 | IC50 | 2 | — | |
HUKGACBEOZARIH
|
6.7 | IC50 | 2 | — | |
JVAFTPDILUBIGR
|
6.7 | IC50 | 7 | — | |
KDJGCVHPUMHUOL
|
6.7 | Ki | 11 | — | |
NGFGTMFVWSDFPS
|
6.7 | IC50 | 32 | — | |
PKULMPKZJZFMMT
|
6.7 | IC50 | 5 | — | |
RWEQMFPLXZZYJD
|
6.7 | IC50 | 5 | — | |
WQQQJDAMPWMJLM
|
6.7 | IC50 | 2 | — | |
MSSYEZHHVYFPOJ
|
6.7 | IC50 | 2 | — | |
AYCPARAPKDAOEN
|
6.7 | Kd | 73 | — | |
IITXSCOJPQUGAM
|
6.7 | IC50 | 2 | — | |
LPTXJCNHKKMGKH
|
6.7 | IC50 | 4 | — | |
SVWXCDGHUFRGHG
|
6.7 | IC50 | 2 | — | |
WXUJAQBSBZLVEV
|
6.7 | IC50 | 3 | Yes | |
ZGZKTZCGFRZSSF
|
6.7 | IC50 | 2 | — | |
DNQMUTHLLWZCPG
|
6.7 | IC50 | 4 | — | |
CPMQDKJELBGISQ
|
6.7 | IC50 | 2 | — | |
KOXCJDZBHOTQQJ
|
6.7 | IC50 | 2 | — | |
RSXAOLHSBWCGJD
|
6.7 | IC50 | 5 | — | |
UZEICMNTLHFXNT
|
6.7 | IC50 | 2 | — | |
PIELNOLQJZOXMR
|
6.7 | IC50 | 2 | — | |
AUBFUJKOXVNDOA
|
6.6 | IC50 | 2 | — | |
GTAMSBNOMFMGCE
|
6.6 | IC50 | 5 | — | |
OJWDCZJTYJWNLF
|
6.6 | IC50 | 2 | — | |
QHQBMNXWJUAAHX
|
6.6 | IC50 | 2 | — | |
WMACZWSUUNMRLW
|
6.6 | IC50 | 2 | — | |
SMPPSGXPGZSJCP
|
6.6 | IC50 | 5 | — | |
YFBPGSDPFRCNOY
|
6.6 | IC50 | 2 | — | |
YXXZXFHNQPWLAW
|
6.6 | IC50 | 2 | — | |
CAJABNJZFXQFQH
|
6.6 | IC50 | 2 | — | |
LFRLUVCEFWYSFT
|
6.6 | IC50 | 2 | — | |
NDHIKTIBSHPKAT
|
6.6 | IC50 | 2 | — | |
PVBVIAFRUDDPSI
|
6.6 | IC50 | 4 | — | |
RZEPRPGFGRQXDI
|
6.6 | IC50 | 3 | — | |
SMPPSGXPGZSJCP
|
6.6 | IC50 | 8 | — |