Target Details
| UniProt AC | O14744 |
|---|---|
| Gene Symbol | PRMT5 |
| Protein Name | Protein arginine N-methyltransferase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05185 (PRMT5) PF17286 (PRMT5_C) PF17285 (PRMT5_TIM) |
Summary
- Multi-target molecules 1,752
- Clinical molecules 0
- Avg pChEMBL 6.86
Active Molecules (1,752)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PNSSQUBIOFAMCO
|
7.5 | IC50 | 2 | — | |
TVXOGQOUJUVEJY
|
7.5 | IC50 | 2 | — | |
WPWTYQBLLPEVPT
|
7.5 | IC50 | 2 | — | |
XGUVQQDNSWJOSM
|
7.5 | IC50 | 2 | — | |
YDRXMXBVUOAKIC
|
7.5 | IC50 | 2 | — | |
ZHQYSBNQTHOGQJ
|
7.5 | IC50 | 2 | — | |
ZKXZLIFRWWKZRY
|
7.5 | IC50 | 2 | — | |
SSNBXGFUCGOVPH
|
7.5 | IC50 | 2 | — | |
WCAILBPALGCSKN
|
7.5 | IC50 | 2 | — | |
QVIQNFYEKFSULJ
|
7.5 | IC50 | 2 | — | |
SPHDXOYHPFKCHP
|
7.5 | IC50 | 2 | — | |
KCFDVNIFNJKLJL
|
7.5 | IC50 | 2 | — | |
HHFHJTNECFJVEY
|
7.5 | IC50 | 2 | — | |
HTFHGNJHNIVONH
|
7.5 | IC50 | 2 | — | |
MJGBOABPPBBMIN
|
7.5 | IC50 | 2 | — | |
WZLWNTDFFZBDCR
|
7.5 | IC50 | 2 | — | |
KCYBVBFDBNEAFQ
|
7.5 | IC50 | 2 | — | |
BTFOMGQKXSAIAQ
|
7.5 | IC50 | 2 | — | |
KKZYAGDKIAWYCA
|
7.5 | IC50 | 2 | — | |
VSJFIITUGWKHFK
|
7.5 | IC50 | 2 | — | |
ZARYNAIOYISPCO
|
7.5 | IC50 | 2 | — | |
CKKMNPIZOMJYSX
|
7.5 | IC50 | 2 | — | |
PFLMLTFIZDNHRL
|
7.5 | IC50 | 2 | — | |
RERIOYBALRXMSF
|
7.5 | IC50 | 2 | — | |
FAAHGTZEAKFSIZ
|
7.4 | IC50 | 2 | — | |
GGRATVWMSFTUKP
|
7.4 | IC50 | 2 | — | |
FYMSRNVGXAVFQT
|
7.4 | IC50 | 2 | — | |
IAEWRKBKPYNKGE
|
7.4 | IC50 | 2 | — | |
KNUIGDFMINUNHZ
|
7.4 | IC50 | 2 | — | |
RDTXSYQRBOBLFV
|
7.4 | IC50 | 2 | — | |
BPTYWAYMKBEXES
|
7.4 | IC50 | 2 | — | |
FSFXOECGEBCOMF
|
7.4 | IC50 | 2 | — | |
OVZNAPQBSKTSCY
|
7.4 | IC50 | 2 | — | |
BDOOKFKZIMWHAH
|
7.4 | IC50 | 2 | — | |
FQCFUAUPXCLTQS
|
7.4 | IC50 | 2 | — | |
ATGRJIJETUETJD
|
7.4 | IC50 | 2 | — | |
BDOGXDDYLRSPFN
|
7.4 | IC50 | 2 | — | |
CFWIOFLDKMVDHR
|
7.4 | IC50 | 2 | — | |
CGYBTANMJBGPQQ
|
7.4 | IC50 | 2 | — | |
FVVBRLOEAZUQPK
|
7.4 | IC50 | 2 | — | |
HVQOUTKOIUZKFP
|
7.4 | IC50 | 2 | — | |
ISROTIMDIBEBDY
|
7.4 | IC50 | 2 | — | |
KFTWJPYJBGSPCN
|
7.4 | IC50 | 2 | — | |
KKOTWRPPUAESJB
|
7.4 | IC50 | 2 | — | |
LUNKLDKBYYSMBI
|
7.4 | IC50 | 2 | — | |
PNKGVHUHKTWGOK
|
7.4 | IC50 | 2 | — | |
MHLOCKTYXIORPC
|
7.4 | IC50 | 2 | — | |
ZRGSHHBXPGVJSR
|
7.4 | IC50 | 2 | — | |
FCYGAQJCBSYGFT
|
7.4 | IC50 | 2 | — | |
VQWMIOJCLWPRMA
|
7.4 | IC50 | 2 | — |