Target Details
| UniProt AC | O14744 |
|---|---|
| Gene Symbol | PRMT5 |
| Protein Name | Protein arginine N-methyltransferase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05185 (PRMT5) PF17286 (PRMT5_C) PF17285 (PRMT5_TIM) |
Summary
- Multi-target molecules 1,752
- Clinical molecules 0
- Avg pChEMBL 6.86
Active Molecules (1,752)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RDJGIPKJLARPSA
|
7.9 | IC50 | 2 | — | |
BDWOIRAPZCUKDY
|
7.8 | IC50 | 2 | — | |
KRXTWDTXDMKVPR
|
7.8 | IC50 | 2 | — | |
ZGYGJQUHLDOYKY
|
7.8 | IC50 | 2 | — | |
AUBWIINMOSIRJK
|
7.8 | IC50 | 2 | — | |
KSGKIKZWGBHRQT
|
7.8 | IC50 | 2 | — | |
OGNJDPSFRGJEAG
|
7.8 | IC50 | 2 | — | |
TVQPEBSGDYZDAP
|
7.8 | IC50 | 2 | — | |
FLZFDCDDLIIXFV
|
7.8 | IC50 | 2 | — | |
LAWDUEFJOJENIJ
|
7.8 | IC50 | 2 | — | |
LUVXBZDRGFIAKS
|
7.8 | IC50 | 2 | — | |
MBXKXQYZJSNKBC
|
7.8 | IC50 | 2 | — | |
OKAFTUQEPQNTET
|
7.8 | IC50 | 2 | — | |
BVCRIZZSQGCZCK
|
7.8 | IC50 | 2 | — | |
GTHDKUZRHRXYTE
|
7.8 | IC50 | 2 | — | |
HZNVSAYIDXARDP
|
7.8 | IC50 | 2 | — | |
RGEFRBMOBQDZBB
|
7.8 | IC50 | 2 | — | |
YUOKSWIONSHHRB
|
7.8 | IC50 | 2 | — | |
ZVCIZCPAJITPQB
|
7.8 | IC50 | 2 | — | |
DNDCXYZRSRFLRY
|
7.8 | IC50 | 2 | — | |
MAQQNBDRZGOONQ
|
7.8 | IC50 | 2 | — | |
XOMOAMNPYQDKPL
|
7.8 | IC50 | 2 | — | |
ZSIWDWYYAHAGDI
|
7.8 | IC50 | 2 | — | |
DUQHYFJHWKPYMW
|
7.8 | IC50 | 2 | — | |
HWWZSLIRECKJAG
|
7.8 | IC50 | 2 | — | |
LVNMCBWIYZNLCV
|
7.8 | IC50 | 2 | — | |
MOENMGQGTQAHPW
|
7.8 | IC50 | 2 | — | |
MQBNHAAEDHNZCH
|
7.8 | IC50 | 2 | — | |
NJWHFGKLLBVQAN
|
7.8 | IC50 | 2 | — | |
WPPYQCCJXGKAGM
|
7.8 | IC50 | 2 | — | |
BRFSSECTMNOADC
|
7.8 | IC50 | 2 | — | |
LPPKXBXXUDNWIG
|
7.8 | IC50 | 2 | — | |
PSNKXGMRHQGRNU
|
7.8 | IC50 | 2 | — | |
PZGSQKASGVWEDK
|
7.8 | IC50 | 2 | — | |
DVZZYZNFLHFCPI
|
7.7 | IC50 | 7 | — | |
XUJMNOQMXWVXQE
|
7.7 | IC50 | 2 | — | |
ZIDCEAFVRIDUJO
|
7.7 | IC50 | 2 | — | |
HQPIJWPBMNFLDK
|
7.7 | IC50 | 2 | — | |
JXFAWTZWNJZBCZ
|
7.7 | IC50 | 2 | — | |
LUVXBZDRGFIAKS
|
7.7 | IC50 | 2 | — | |
PBAIMAKMPCRAON
|
7.7 | IC50 | 2 | — | |
UEQHNRXLIUOJTG
|
7.7 | IC50 | 2 | — | |
VBEGBQCJGDEECI
|
7.7 | IC50 | 2 | — | |
ZGYGJQUHLDOYKY
|
7.7 | IC50 | 2 | — | |
AOSQGWUEZPSSNR
|
7.7 | IC50 | 2 | — | |
HXCQIQYQJHILRY
|
7.7 | IC50 | 2 | — | |
IQOXVADYZAROMQ
|
7.7 | IC50 | 2 | — | |
JUCLHDNTLJBIAI
|
7.7 | IC50 | 2 | — | |
LUVXBZDRGFIAKS
|
7.7 | IC50 | 2 | — | |
NENINCVAVDXELX
|
7.7 | IC50 | 2 | — |