Target Details
| UniProt AC | O14744 |
|---|---|
| Gene Symbol | PRMT5 |
| Protein Name | Protein arginine N-methyltransferase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05185 (PRMT5) PF17286 (PRMT5_C) PF17285 (PRMT5_TIM) |
Summary
- Multi-target molecules 1,752
- Clinical molecules 0
- Avg pChEMBL 6.86
Active Molecules (1,752)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VPIMQKCPFWKIKW
|
8.0 | IC50 | 2 | — | |
VTRYSFDFIFLQHT
|
8.0 | IC50 | 2 | — | |
WAAMFRLMPUTKHA
|
8.0 | IC50 | 2 | — | |
WCUKHIOLFPGARE
|
8.0 | IC50 | 2 | — | |
WGFHENPHGYFRCF
|
8.0 | IC50 | 2 | — | |
WKJFWQDWRXBVAI
|
8.0 | IC50 | 3 | — | |
WKJFWQDWRXBVAI
|
8.0 | IC50 | 3 | — | |
WMKMNMBGLYSSCF
|
8.0 | IC50 | 3 | — | |
WTBCNABVOCLART
|
8.0 | IC50 | 2 | — | |
XKURGPLKALAOMX
|
8.0 | IC50 | 2 | — | |
XONGKOCVDOMGMY
|
8.0 | IC50 | 2 | — | |
XQGUHJKRXPMBEY
|
8.0 | IC50 | 3 | — | |
ZCFKJUKYINQBKY
|
8.0 | IC50 | 3 | — | |
ZGEWUHKMLCRENE
|
8.0 | IC50 | 2 | — | |
ZLSHESUSBQPONM
|
8.0 | IC50 | 3 | — | |
KIKHICGDJZUHBB
|
8.0 | IC50 | 2 | — | |
MZESOICLUQKLAH
|
8.0 | IC50 | 2 | — | |
OOVRTBWZEQWLIY
|
8.0 | IC50 | 2 | — | |
WIPONRQAVGXVBZ
|
8.0 | IC50 | 2 | — | |
AVJDKCLSVKCKCR
|
8.0 | IC50 | 2 | — | |
KYOVWTVYHRQPLL
|
8.0 | IC50 | 2 | — | |
LMQXLKNSRLIXHZ
|
8.0 | IC50 | 2 | — | |
MQBNHAAEDHNZCH
|
8.0 | IC50 | 2 | — | |
PNEWSTDPFYPNQM
|
8.0 | IC50 | 2 | — | |
VFSOQQVDAIJQES
|
8.0 | IC50 | 2 | — | |
LVIBWWLMMYXMBV
|
8.0 | IC50 | 2 | — | |
WFQRQFNZAQBGMH
|
7.9 | IC50 | 2 | — | |
ZYSOFQGKMVBGJG
|
7.9 | IC50 | 2 | — | |
RIIGOQBWTOGALW
|
7.9 | IC50 | 2 | — | |
WMBBADXVRALADZ
|
7.9 | IC50 | 2 | — | |
WSDNGHACVSEGKR
|
7.9 | IC50 | 2 | — | |
KHARBUSEIBEVGF
|
7.9 | IC50 | 2 | — | |
LTPABOINPMWTKU
|
7.9 | IC50 | 3 | — | |
MKFVJVPIFLNNNU
|
7.9 | IC50 | 2 | — | |
NAYGLAGPJBUELD
|
7.9 | IC50 | 2 | — | |
RMCXWGKWLAZNAS
|
7.9 | IC50 | 2 | — | |
WZUPWIUCGGYCAP
|
7.9 | IC50 | 2 | — | |
XUJMNOQMXWVXQE
|
7.9 | IC50 | 2 | — | |
WHXFFFPKVVPLCI
|
7.9 | IC50 | 2 | — | |
LPPKXBXXUDNWIG
|
7.9 | IC50 | 2 | — | |
FAAHGTZEAKFSIZ
|
7.9 | IC50 | 2 | — | |
HTFHGNJHNIVONH
|
7.9 | IC50 | 2 | — | |
LUVXBZDRGFIAKS
|
7.9 | IC50 | 2 | — | |
XGHYOSZCJQLKBG
|
7.9 | IC50 | 2 | — | |
ZGYGJQUHLDOYKY
|
7.9 | IC50 | 2 | — | |
OYQCVGQLLAQRPR
|
7.9 | IC50 | 2 | — | |
FQHZZVSKMGNOFN
|
7.9 | IC50 | 2 | — | |
LNSLBEXUTPFUMW
|
7.9 | IC50 | 2 | — | |
IPYAEANWZBKIHO
|
7.9 | IC50 | 2 | — | |
NZQLESMZWHEEBK
|
7.9 | IC50 | 2 | — |