Target Details
| UniProt AC | O14744 |
|---|---|
| Gene Symbol | PRMT5 |
| Protein Name | Protein arginine N-methyltransferase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05185 (PRMT5) PF17286 (PRMT5_C) PF17285 (PRMT5_TIM) |
Summary
- Multi-target molecules 1,752
- Clinical molecules 0
- Avg pChEMBL 6.86
Active Molecules (1,752)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DTFULKURTJXYSJ
|
8.0 | IC50 | 2 | — | |
DWKQTUXGXSWCDD
|
8.0 | IC50 | 3 | — | |
FEAJNCPPXMPQES
|
8.0 | IC50 | 3 | — | |
GBVXGNTZYNSJEA
|
8.0 | IC50 | 2 | — | |
GPFBMASCYPSJBO
|
8.0 | IC50 | 2 | — | |
GVJMFHDJGPYKLA
|
8.0 | IC50 | 3 | — | |
HGUYPPYOIOGKSD
|
8.0 | IC50 | 2 | — | |
HJXJQDDRWMMLCV
|
8.0 | IC50 | 3 | — | |
HMABXZUBNVAHQP
|
8.0 | IC50 | 2 | — | |
HMABXZUBNVAHQP
|
8.0 | IC50 | 2 | — | |
HPBVVJIUOMEVGS
|
8.0 | IC50 | 2 | — | |
HTCLDNGTQXWAJI
|
8.0 | IC50 | 2 | — | |
ILLCLAICZDCVEL
|
8.0 | IC50 | 2 | — | |
IURSMTTZFIKUIM
|
8.0 | IC50 | 2 | — | |
IVTMJHXAJSJIJB
|
8.0 | IC50 | 3 | — | |
IXIDISRBMSVZIR
|
8.0 | IC50 | 2 | — | |
JBSJNGSDWNLQEA
|
8.0 | IC50 | 3 | — | |
JZIQSLJXRARYPS
|
8.0 | IC50 | 3 | — | |
KBGVQKBVRSHTTD
|
8.0 | IC50 | 3 | — | |
KHBGXDWIVZWUNL
|
8.0 | IC50 | 2 | — | |
KIXGVMKUHVKGID
|
8.0 | IC50 | 2 | — | |
LPPKXBXXUDNWIG
|
8.0 | IC50 | 2 | — | |
LXLHIUQPFNWAHW
|
8.0 | IC50 | 2 | — | |
MCQVQEZKVZPHFA
|
8.0 | IC50 | 2 | — | |
MEEWZBXFBKLDQW
|
8.0 | IC50 | 3 | — | |
MESYGUCCDFFLBX
|
8.0 | IC50 | 3 | — | |
MNSWNMQWUYUILS
|
8.0 | IC50 | 2 | — | |
NLUQVZVYDAYLMT
|
8.0 | IC50 | 2 | — | |
OOVWVMNOAHXDHJ
|
8.0 | IC50 | 3 | — | |
PKDWWYHNKYEKTE
|
8.0 | IC50 | 2 | — | |
PMPGBDNVPYTVPO
|
8.0 | IC50 | 3 | — | |
PNBXLWISZBWELN
|
8.0 | IC50 | 2 | — | |
PYOFHQAYYVSQRU
|
8.0 | IC50 | 2 | — | |
QGYDWGDOUSDHOL
|
8.0 | IC50 | 2 | — | |
QKXCKYWFVOINKB
|
8.0 | IC50 | 2 | — | |
QSAIZEODNWGRTL
|
8.0 | IC50 | 2 | — | |
QWUFPKCHLDECDK
|
8.0 | IC50 | 3 | — | |
RHUDVSFXQKAJPK
|
8.0 | IC50 | 3 | — | |
RSBRQRLAIMVFQM
|
8.0 | IC50 | 2 | — | |
RXIBZUMVYIXZGT
|
8.0 | IC50 | 2 | — | |
RYYVQIAUSPYHKR
|
8.0 | IC50 | 2 | — | |
SJACEMSZVUVEEJ
|
8.0 | IC50 | 2 | — | |
TYNZPVIHFRFFIF
|
8.0 | IC50 | 2 | — | |
TZELHXQLVZPLPQ
|
8.0 | IC50 | 2 | — | |
UDWLJIOTNBATOE
|
8.0 | IC50 | 2 | — | |
UEPOZFJIJCXOLS
|
8.0 | IC50 | 2 | — | |
USKRIRBSNVMSTN
|
8.0 | IC50 | 3 | — | |
UTFXTWOXDJLLLY
|
8.0 | IC50 | 3 | — | |
VFURLHFFODVRHZ
|
8.0 | IC50 | 3 | — | |
VJKMQGVETATWJV
|
8.0 | IC50 | 2 | — |