Target Details
| UniProt AC | O14744 |
|---|---|
| Gene Symbol | PRMT5 |
| Protein Name | Protein arginine N-methyltransferase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05185 (PRMT5) PF17286 (PRMT5_C) PF17285 (PRMT5_TIM) |
Summary
- Multi-target molecules 1,752
- Clinical molecules 0
- Avg pChEMBL 6.86
Active Molecules (1,752)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZSMBTEMKYUTYOD
|
8.2 | IC50 | 2 | — | |
AAXSOKYDKLFULN
|
8.2 | IC50 | 2 | — | |
FDGJEHIDEQYOOR
|
8.2 | IC50 | 2 | — | |
UMSBLTPKMWVNEW
|
8.2 | IC50 | 2 | — | |
VSJFIITUGWKHFK
|
8.2 | IC50 | 2 | — | |
MLHRTWKNJOQXHD
|
8.2 | IC50 | 2 | — | |
DOBNWPZLHQEPBQ
|
8.2 | IC50 | 2 | — | |
GIVBMSCEMGCGQJ
|
8.2 | IC50 | 2 | — | |
SVLUJONIVKIVAX
|
8.2 | IC50 | 2 | — | |
WNNVPFLHXIDGHS
|
8.2 | IC50 | 2 | — | |
LVIBWWLMMYXMBV
|
8.2 | IC50 | 2 | — | |
YKZDTNIWDJJWMK
|
8.2 | IC50 | 2 | — | |
XINDTHWOOIIELL
|
8.2 | IC50 | 2 | — | |
YXURNYCBOAWPHP
|
8.2 | IC50 | 2 | — | |
BNRVKYALGCENTO
|
8.1 | IC50 | 2 | — | |
BNNBXFJEDQYISJ
|
8.1 | IC50 | 2 | — | |
OGKDUZCIRBBSNS
|
8.1 | IC50 | 2 | — | |
RTYLGFBFEFKSEE
|
8.1 | IC50 | 2 | — | |
NWCCQRMIKQRTFW
|
8.1 | IC50 | 2 | — | |
UNJFWYGMXNSASF
|
8.1 | IC50 | 2 | — | |
ADMXDABBLUUEPG
|
8.1 | IC50 | 2 | — | |
ZTTUACZVEKPJNE
|
8.1 | IC50 | 2 | — | |
FQCFUAUPXCLTQS
|
8.1 | IC50 | 2 | — | |
LAEYVCMVWKYXNL
|
8.1 | IC50 | 2 | — | |
MHGLIAYUKWFWGJ
|
8.1 | IC50 | 2 | — | |
OSOFWQCHKHEEPX
|
8.1 | IC50 | 2 | — | |
HOLKSORSINFXCU
|
8.1 | IC50 | 2 | — | |
IAKJMOBYLLVGKR
|
8.1 | IC50 | 2 | — | |
VFSOQQVDAIJQES
|
8.1 | IC50 | 2 | — | |
XGHYOSZCJQLKBG
|
8.1 | IC50 | 2 | — | |
MWFLCEUDWRURTE
|
8.1 | IC50 | 2 | — | |
YAKKCODNQDUTDD
|
8.1 | IC50 | 2 | — | |
CATWWGFETIUKQV
|
8.1 | IC50 | 2 | — | |
UNJFWYGMXNSASF
|
8.1 | IC50 | 2 | — | |
LGXJELYWRWBUQZ
|
8.0 | IC50 | 2 | — | |
YVVQZOCDTONFOY
|
8.0 | IC50 | 2 | — | |
GAFFRVOQKBCJAR
|
8.0 | IC50 | 2 | — | |
JLCCNYVTIWRPIZ
|
8.0 | IC50 | 2 | — | |
LPPKXBXXUDNWIG
|
8.0 | IC50 | 2 | — | |
WWOOWAHTEXIWBO
|
8.0 | IC50 | 2 | — | |
SOWWMZNHUAHSIN
|
8.0 | IC50 | 2 | — | |
AXJQYJGKIJOWPN
|
8.0 | IC50 | 3 | — | |
BIAXKEIJSOITHA
|
8.0 | IC50 | 3 | — | |
BTVPTMWTKQPMRW
|
8.0 | IC50 | 3 | — | |
COEGFZLXABUQEE
|
8.0 | IC50 | 2 | — | |
CSANZLJSAQBTMB
|
8.0 | IC50 | 2 | — | |
CYZOLNVYTJFHLM
|
8.0 | IC50 | 3 | — | |
CZQDXGWPFGVYEA
|
8.0 | IC50 | 2 | — | |
DMOUDASMWZDGHT
|
8.0 | IC50 | 2 | — | |
DRJLIJVRIGWPPF
|
8.0 | IC50 | 3 | — |