Target Details
| UniProt AC | O14744 |
|---|---|
| Gene Symbol | PRMT5 |
| Protein Name | Protein arginine N-methyltransferase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05185 (PRMT5) PF17286 (PRMT5_C) PF17285 (PRMT5_TIM) |
Summary
- Multi-target molecules 1,752
- Clinical molecules 0
- Avg pChEMBL 6.86
Active Molecules (1,752)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SYQNLTRPVHTWDK
|
8.7 | IC50 | 2 | — | |
DVYGIYCMNUKVBE
|
8.7 | IC50 | 2 | — | |
NYDWXLPQKNNOER
|
8.7 | IC50 | 2 | — | |
OYPQTNGMDHACTQ
|
8.7 | IC50 | 2 | — | |
FXUVRIZNKOANNW
|
8.6 | IC50 | 2 | — | |
KFTWIUQJWMRJQW
|
8.6 | IC50 | 2 | — | |
QSWFOYVXGNRPRC
|
8.6 | IC50 | 2 | — | |
HVVYGSDCWYHXPY
|
8.6 | IC50 | 2 | — | |
AGOIKKPEOPSIHC
|
8.6 | IC50 | 2 | — | |
QIEPEOWPAMHREL
|
8.6 | IC50 | 2 | — | |
LPPKXBXXUDNWIG
|
8.6 | IC50 | 2 | — | |
IXCWXYLRELEGRS
|
8.6 | IC50 | 2 | — | |
LLWQXCUVFNXITH
|
8.6 | IC50 | 2 | — | |
YNNRDSIFCSVIDD
|
8.6 | IC50 | 2 | — | |
PIERCIOPKDBMLC
|
8.5 | IC50 | 2 | — | |
KSXBQFKWCCJWNH
|
8.5 | IC50 | 2 | — | |
LKKYUVKLMITZGD
|
8.5 | IC50 | 2 | — | |
NOWWVBFXXUUWKN
|
8.5 | IC50 | 2 | — | |
UEAAYHPSDGGRQI
|
8.5 | IC50 | 2 | — | |
NZHNTAQIEXXLET
|
8.5 | IC50 | 2 | — | |
MCCXVFKEWSFETL
|
8.5 | IC50 | 2 | — | |
OWCCWTKMNKIDAJ
|
8.5 | IC50 | 2 | — | |
XDSGZKIAGNIVDK
|
8.5 | IC50 | 2 | — | |
TWPCXFCEZJPTDU
|
8.5 | IC50 | 2 | — | |
YFBYFUIGKMIFGW
|
8.4 | IC50 | 2 | — | |
BQXHUBIROWQFCN
|
8.4 | IC50 | 2 | — | |
NSYXJLZEQPXXPZ
|
8.4 | IC50 | 2 | — | |
ZYHQRCUTLQBIMQ
|
8.4 | IC50 | 2 | — | |
ITEKIFMGFZAFPM
|
8.4 | IC50 | 2 | — | |
FAKDLANDAFIUOS
|
8.4 | IC50 | 2 | — | |
SVJLKRXTYXVBPP
|
8.4 | IC50 | 2 | — | |
TWKYXZSXXXKKJU
|
8.4 | IC50 | 2 | — | |
FAAHGTZEAKFSIZ
|
8.3 | IC50 | 2 | — | |
KFFJVMZXYDPIDQ
|
8.3 | IC50 | 2 | — | |
LVIBWWLMMYXMBV
|
8.3 | IC50 | 2 | — | |
FFQLPKBDTZBCDL
|
8.3 | IC50 | 2 | — | |
MLESHNTYCKAIOZ
|
8.3 | IC50 | 2 | — | |
QWEACAUAEFHICR
|
8.3 | IC50 | 2 | — | |
WFQRQFNZAQBGMH
|
8.3 | IC50 | 2 | — | |
ROBDUKXVDWAJJB
|
8.3 | IC50 | 2 | — | |
RFOSOYYKBITPCA
|
8.3 | IC50 | 2 | — | |
NXXBDYHMHHINFC
|
8.3 | Ki | 2 | — | |
CKDKKHTYJFBKPI
|
8.2 | IC50 | 2 | — | |
WGKVJYZNSMWPLN
|
8.2 | IC50 | 2 | — | |
JWZDBSDWWKOHJH
|
8.2 | IC50 | 2 | — | |
QMOPRHVNRMKVLE
|
8.2 | IC50 | 2 | — | |
BJIUKEMXFQJDBZ
|
8.2 | IC50 | 2 | — | |
HQPPFCPKICDTKJ
|
8.2 | IC50 | 2 | — | |
SKLDQNBOLVKBJG
|
8.2 | IC50 | 2 | — | |
SEAKHLUQEKBMJL
|
8.2 | IC50 | 2 | — |