Target Details
| UniProt AC | O14744 |
|---|---|
| Gene Symbol | PRMT5 |
| Protein Name | Protein arginine N-methyltransferase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05185 (PRMT5) PF17286 (PRMT5_C) PF17285 (PRMT5_TIM) |
Summary
- Multi-target molecules 1,752
- Clinical molecules 0
- Avg pChEMBL 6.86
Active Molecules (1,752)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IQAXJVBGIYHEKZ
|
7.0 | IC50 | 2 | — | |
IVBZHEINLFUIQJ
|
7.0 | IC50 | 3 | — | |
JAQUJSJEKOIKMG
|
7.0 | IC50 | 2 | — | |
JIGZQWHXOPRBAM
|
7.0 | IC50 | 2 | — | |
JPWCFWRCXQIJQU
|
7.0 | IC50 | 2 | — | |
KDNZXPIBYGLZSF
|
7.0 | IC50 | 3 | — | |
KRVUJADOXCFNQH
|
7.0 | IC50 | 3 | — | |
KSQRQFILPJBFOD
|
7.0 | IC50 | 2 | — | |
KSYRPYAWNHUPGY
|
7.0 | IC50 | 3 | — | |
LARDAUCPJGBKQE
|
7.0 | IC50 | 2 | — | |
LFAAXEJCOZHVLW
|
7.0 | IC50 | 3 | — | |
LGHQSFKSGYAABV
|
7.0 | IC50 | 4 | — | |
LRIBFTQSIQVDGH
|
7.0 | IC50 | 2 | — | |
LUOQYHYFHBUMIB
|
7.0 | IC50 | 2 | — | |
LXPVDWMKUGIWPI
|
7.0 | IC50 | 2 | — | |
MGGYNFAYGPUCEJ
|
7.0 | IC50 | 3 | — | |
MJRJZLPWTTYBFJ
|
7.0 | IC50 | 2 | — | |
MKDMZRDYSAYRKH
|
7.0 | IC50 | 3 | — | |
MLWSIQHUCSUOHY
|
7.0 | IC50 | 2 | — | |
MUEFQHSUCVGKRN
|
7.0 | IC50 | 2 | — | |
NECXRLQHYLEXMB
|
7.0 | IC50 | 2 | — | |
NMJAYJXRBDEREO
|
7.0 | IC50 | 3 | — | |
NWHQEODZVXCGLE
|
7.0 | IC50 | 2 | — | |
NXVSYULUHFMNFS
|
7.0 | IC50 | 2 | — | |
NZRSCPPEGJHBCC
|
7.0 | IC50 | 2 | — | |
ODQLHMKBCVSSON
|
7.0 | IC50 | 3 | — | |
OHQMWDFBWCSXPT
|
7.0 | IC50 | 3 | — | |
OMWNBKRKLVGYCB
|
7.0 | IC50 | 2 | — | |
OPTWLYCKKBTKGQ
|
7.0 | IC50 | 2 | — | |
PDECWAXDIYOBDH
|
7.0 | IC50 | 2 | — | |
PLQIBMXOODUJNH
|
7.0 | IC50 | 3 | — | |
PPVMVYKPZIPBCR
|
7.0 | IC50 | 2 | — | |
PPYDCTMHTZSRFS
|
7.0 | IC50 | 2 | — | |
PVULNZOSBJJNKR
|
7.0 | IC50 | 2 | — | |
PXBMUZZEWGRRFH
|
7.0 | IC50 | 2 | — | |
PXOAPOFERXXQCH
|
7.0 | IC50 | 2 | — | |
PYJYPCQUPPXWKE
|
7.0 | IC50 | 2 | — | |
QDGVXHDUIARDED
|
7.0 | IC50 | 2 | — | |
QQGBVSSFUYPMPW
|
7.0 | IC50 | 2 | — | |
QYKICPAUVKJFKV
|
7.0 | IC50 | 2 | — | |
RHLCHYYLKCLXKV
|
7.0 | IC50 | 2 | — | |
RUOYVUIAMGFNRH
|
7.0 | IC50 | 2 | — | |
SEEZEQABSNHWCW
|
7.0 | IC50 | 2 | — | |
SGZGEEKSSZABMR
|
7.0 | IC50 | 2 | — | |
SPLZQUBXMVIDDQ
|
7.0 | IC50 | 3 | — | |
SSWPJPJGDIEQNJ
|
7.0 | IC50 | 2 | — | |
UCVJQBJYLYMFCI
|
7.0 | IC50 | 2 | — | |
UGMFITXTVCKADG
|
7.0 | IC50 | 2 | — | |
UJNGAUOMUFLAKY
|
7.0 | IC50 | 2 | — | |
VTJXGUKIIWTSQP
|
7.0 | IC50 | 3 | — |