Target Details
| UniProt AC | O14744 |
|---|---|
| Gene Symbol | PRMT5 |
| Protein Name | Protein arginine N-methyltransferase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05185 (PRMT5) PF17286 (PRMT5_C) PF17285 (PRMT5_TIM) |
Summary
- Multi-target molecules 1,752
- Clinical molecules 0
- Avg pChEMBL 6.86
Active Molecules (1,752)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KTCOIPWPIIWIHW
|
7.1 | IC50 | 2 | — | |
MJXMAOIXWZBANA
|
7.1 | IC50 | 2 | — | |
OFVDIVGNIWASKX
|
7.1 | IC50 | 2 | — | |
COKWWTMKYXNVKU
|
7.0 | Kd | 2 | — | |
FWLIDJVSTVQPSU
|
7.0 | IC50 | 2 | — | |
OKWBLHUSYOVGDB
|
7.0 | IC50 | 2 | — | |
QRDWYENEHGIBNI
|
7.0 | IC50 | 2 | — | |
VAEAPPUJJADYEH
|
7.0 | IC50 | 2 | — | |
XOIOLGWPWCUMRV
|
7.0 | IC50 | 2 | — | |
BWMOUMPYKNMECB
|
7.0 | IC50 | 2 | — | |
FHACYTRKYWYOHP
|
7.0 | IC50 | 2 | — | |
WFXAZZULKQWXBX
|
7.0 | IC50 | 2 | — | |
WMVXWZVXOJHCIR
|
7.0 | IC50 | 2 | — | |
JXLRQFLREJBDHU
|
7.0 | IC50 | 2 | — | |
SCBNTLBKBPTTRW
|
7.0 | IC50 | 2 | — | |
CFIHKSZSFICELW
|
7.0 | IC50 | 2 | — | |
JCBQHEUBFGHFAE
|
7.0 | IC50 | 2 | — | |
VIZNSDUBXAESGA
|
7.0 | IC50 | 2 | — | |
FZTTVOOCSZSXBA
|
7.0 | IC50 | 2 | — | |
HQZPPIJFNGWEMW
|
7.0 | IC50 | 2 | — | |
ACUUAZBXPCUOGH
|
7.0 | IC50 | 2 | — | |
AGYPZLZLPAXHPC
|
7.0 | IC50 | 2 | — | |
AHSCEIIJIDWUSO
|
7.0 | IC50 | 3 | — | |
ARQMZHUCEQVMBR
|
7.0 | IC50 | 3 | — | |
BBPXWJIFZIZQJN
|
7.0 | IC50 | 3 | — | |
BOBUAHFIFWJQLJ
|
7.0 | IC50 | 2 | — | |
BSCNZRRBABACDM
|
7.0 | IC50 | 3 | — | |
BSVGKYJBSHYMPI
|
7.0 | IC50 | 2 | — | |
BUYPRXDEARMMOQ
|
7.0 | IC50 | 2 | — | |
CHGOOLWBTBPORO
|
7.0 | IC50 | 2 | — | |
CNMMZTWHDXVNBY
|
7.0 | IC50 | 2 | — | |
CPJMLOLDZRVYHI
|
7.0 | IC50 | 3 | — | |
DHFFBRYFHFPZFD
|
7.0 | IC50 | 3 | — | |
DMTXVXQTQRVQHI
|
7.0 | IC50 | 3 | — | |
DMTXVXQTQRVQHI
|
7.0 | IC50 | 2 | — | |
DRJLIJVRIGWPPF
|
7.0 | IC50 | 3 | — | |
FHQSJSBYVAKWRU
|
7.0 | IC50 | 2 | — | |
FILHFTADVJSLHJ
|
7.0 | IC50 | 2 | — | |
FQCUFTGCWIMALT
|
7.0 | IC50 | 3 | — | |
FVRYRJCXQJJQGW
|
7.0 | IC50 | 2 | — | |
FWOOHCKJEYAWAX
|
7.0 | IC50 | 2 | — | |
FZMXQSIAXDAVST
|
7.0 | IC50 | 2 | — | |
GPZIVZOMXUPDAH
|
7.0 | IC50 | 2 | — | |
GSYMIZCPPWKOMJ
|
7.0 | IC50 | 2 | — | |
GTDKKNHZRPOBLP
|
7.0 | IC50 | 3 | — | |
HAUIGOXTLZUKNI
|
7.0 | IC50 | 2 | — | |
HCRXVBCEXCJJSV
|
7.0 | IC50 | 2 | — | |
HNQUMERETQBILG
|
7.0 | IC50 | 2 | — | |
IHDQTTUADPDHJK
|
7.0 | IC50 | 3 | — | |
IIERSVJQEGSVFW
|
7.0 | IC50 | 2 | — |