Target Details
| UniProt AC | O14744 |
|---|---|
| Gene Symbol | PRMT5 |
| Protein Name | Protein arginine N-methyltransferase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05185 (PRMT5) PF17286 (PRMT5_C) PF17285 (PRMT5_TIM) |
Summary
- Multi-target molecules 1,752
- Clinical molecules 0
- Avg pChEMBL 6.86
Active Molecules (1,752)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YEADOMAJOBBXBU
|
10.3 | Ki | 2 | — | |
IFXCLMGNYHEINP
|
9.7 | IC50 | 2 | — | |
IUBFXROFEOCTGQ
|
9.7 | IC50 | 3 | — | |
XXYWLEVHJQGNLG
|
9.7 | IC50 | 2 | — | |
DBSMLQTUDJVICQ
|
9.6 | IC50 | 2 | — | |
SJVIZOJFYFICDC
|
9.5 | IC50 | 2 | — | |
WJEGMAZWBVSDGG
|
9.5 | IC50 | 2 | — | |
WSUFOFSXVANLHU
|
9.4 | IC50 | 2 | — | |
YUKZPONUUIFCET
|
9.4 | IC50 | 2 | — | |
CDHNSYFOBQQCHE
|
9.4 | IC50 | 2 | — | |
OQFRQLWUXSTHHK
|
9.4 | IC50 | 3 | — | |
PMLVTAUALHGTDV
|
9.4 | IC50 | 2 | — | |
QRIOWSCVJSHXMY
|
9.4 | IC50 | 2 | — | |
JZXUWFPUMKZMTA
|
9.3 | IC50 | 2 | — | |
HUEIOZOSEXCRNL
|
9.2 | IC50 | 2 | — | |
BSFFOCFGPQDGGM
|
9.2 | IC50 | 2 | — | |
XOAGRGZQXSOUHH
|
9.2 | IC50 | 2 | — | |
KVWKXLFUYJHPJV
|
9.2 | IC50 | 2 | — | |
KCLDZPHNBLIJFB
|
9.2 | IC50 | 2 | — | |
YBNXLYGCTDZHSG
|
9.2 | IC50 | 2 | — | |
LITUSLGKCXVKPY
|
9.1 | IC50 | 2 | — | |
VCECDMPBGSDIQI
|
9.1 | IC50 | 2 | — | |
WNAZWXPYATUMBE
|
9.1 | IC50 | 2 | — | |
CQOJYBCVEDQRIV
|
9.1 | IC50 | 2 | — | |
DFICHQMERPRTQC
|
9.1 | IC50 | 2 | — | |
XNAPHTQOZUJCQT
|
9.1 | IC50 | 2 | — | |
BEWFVLYVAWLKQZ
|
9.1 | IC50 | 2 | — | |
IWKRBGVYEYVENH
|
9.1 | IC50 | 2 | — | |
XGNCIUCSKJERPK
|
9.1 | IC50 | 2 | — | |
BKXOWBKZDGTLFX
|
9.0 | IC50 | 2 | — | |
GTCYWLXMJRCJNE
|
9.0 | IC50 | 2 | — | |
HADKMWKTGHTOQQ
|
9.0 | IC50 | 2 | — | |
HBGHQRGHFNTSDP
|
9.0 | IC50 | 2 | — | |
IXQKPZSMAFSERF
|
9.0 | IC50 | 2 | — | |
WZVHNCLDXMIBSL
|
9.0 | IC50 | 2 | — | |
XLDLIFBOVZRYMG
|
9.0 | IC50 | 2 | — | |
YDGIDMHKHFFVPX
|
9.0 | IC50 | 2 | — | |
YPLNCUPFAOBMQF
|
9.0 | IC50 | 2 | — | |
ARLUXFUKOHIWIA
|
9.0 | IC50 | 2 | — | |
MURBFVDKWOUNSQ
|
8.9 | IC50 | 2 | — | |
FJWSDBIMYNCUBC
|
8.8 | IC50 | 2 | — | |
NRHGITZZOBOACN
|
8.8 | IC50 | 2 | — | |
BHVYMDWQWQIEBZ
|
8.8 | IC50 | 2 | — | |
HKXVKNIGULOIGM
|
8.8 | IC50 | 2 | — | |
NVZVVFMXEHOMQR
|
8.8 | IC50 | 2 | — | |
BDWOIRAPZCUKDY
|
8.8 | IC50 | 2 | — | |
HLGUJTSUABXTJI
|
8.8 | IC50 | 2 | — | |
JZUYFQWEDPPVCE
|
8.8 | IC50 | 2 | — | |
KQQVFXIBOQCHBA
|
8.7 | IC50 | 2 | — | |
RPTKDLSRYWBUPV
|
8.7 | IC50 | 2 | — |