Target Details
| UniProt AC | O14730 |
|---|---|
| Gene Symbol | RIOK3 |
| Protein Name | Serine/threonine-protein kinase RIO3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01163 (RIO1) |
Summary
- Multi-target molecules 16
- Clinical molecules 8
- Avg pChEMBL 6.7
Active Molecules (16)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UIARLYUEJFELEN
|
8.1 | Kd | 289 | Yes | |
XZXHXSATPCNXJR
|
7.4 | Kd | 165 | Yes | |
YYLKKYCXAOBSRM
|
7.2 | Kd | 191 | — | |
HKSZLNNOFSGOKW
|
7.1 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
7.1 | Kd | 213 | — | |
JOOXLOJCABQBSG
|
7.0 | Kd | 139 | — | |
NHHQJBCNYHBUSI
|
6.7 | Kd | 220 | — | |
UCBIQZUJJSVQHL
|
6.5 | Kd | 8 | — | |
OYONTEXKYJZFHA
|
6.4 | Kd | 69 | Yes | |
BMGQWWVMWDBQGC
|
6.4 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.4 | Kd | 91 | Yes | |
GCIKSSRWRFVXBI
|
6.2 | Kd | 109 | Yes | |
ZCBUQCWBWNUWSU
|
6.2 | Kd | 59 | — | |
BPNUQXPIQBZCMR
|
6.2 | Kd | 83 | Yes | |
PIQCTGMSNWUMAF
|
6.2 | Kd | 137 | Yes | |
RITAVMQDGBJQJZ
|
6.0 | Kd | 43 | — |