Target Details
| UniProt AC | O14672 |
|---|---|
| Gene Symbol | ADAM10 |
| Protein Name | Disintegrin and metalloproteinase domain-containing protein 10 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21299 (ADAM10_Cys-rich) PF00200 (Disintegrin) PF13574 (Reprolysin_2) |
Summary
- Multi-target molecules 111
- Clinical molecules 78
- Avg pChEMBL 7.16
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (111)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AZEKZZSSVLIPCQ
|
6.4 | Ki | 2 | — | |
ONHHOEXQJXSXKC
|
6.3 | IC50 | 2 | — | |
QVNZBDLTUKCPGJ
|
6.3 | IC50 | 10 | — | |
ANOPQMHOFNTJCB
|
6.3 | IC50 | 4 | Yes | |
HJLAUHYNMNIAAR
|
6.3 | IC50 | 2 | — | |
BXLWVAKSQMYQKF
|
6.2 | Ki | 5 | Yes | |
KALKLNBLKRHXMI
|
6.1 | IC50 | 2 | — | |
LRRAUDSVXJEODP
|
6.1 | Ki | 6 | Yes | |
BSIZUMJRKYHEBR
|
6.0 | IC50 | 15 | Yes | |
GHBQSNPRMVUGFE
|
6.0 | IC50 | 2 | — | |
BQDVTMRZPWSYOT
|
6.0 | IC50 | 7 | — |