Target Details
| UniProt AC | O14672 |
|---|---|
| Gene Symbol | ADAM10 |
| Protein Name | Disintegrin and metalloproteinase domain-containing protein 10 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21299 (ADAM10_Cys-rich) PF00200 (Disintegrin) PF13574 (Reprolysin_2) |
Summary
- Multi-target molecules 111
- Clinical molecules 78
- Avg pChEMBL 7.16
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (111)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JRJYBZYDJRBFTK
|
7.2 | IC50 | 3 | Yes | |
GYKATPWJHDSXEC
|
7.2 | IC50 | 4 | Yes | |
JQTQTEMWCRRECT
|
7.2 | IC50 | 3 | Yes | |
RAJATBMMJHSJNJ
|
7.2 | IC50 | 3 | Yes | |
MAVDNGWEBZTACC
|
7.2 | IC50 | 9 | Yes | |
MAVDNGWEBZTACC
|
7.2 | IC50 | 6 | — | |
ZQQITVPPJYESAU
|
7.1 | Ki | 3 | — | |
REAAGXUAXYMPTM
|
7.1 | IC50 | 5 | Yes | |
VOGZLMQCZGOADJ
|
7.1 | IC50 | 3 | Yes | |
YCCUTKPNUYYNML
|
7.1 | IC50 | 3 | Yes | |
YDJAXPJDHWQNLF
|
7.1 | IC50 | 3 | Yes | |
DSPHOALBCOPTJE
|
7.1 | IC50 | 3 | Yes | |
IWKMSLYRBYXTNT
|
7.1 | IC50 | 3 | Yes | |
XYYDUHNDMZDPKL
|
7.1 | IC50 | 3 | Yes | |
OEHDRCQWQWUTCW
|
7.1 | IC50 | 2 | — | |
UCFPOZCPIVOGIJ
|
7.1 | IC50 | 2 | — | |
MAXWOEDRRCSRHI
|
7.0 | IC50 | 3 | Yes | |
HJNKYGBTSGQBDU
|
7.0 | IC50 | 10 | — | |
XKPUKZQRNSFQLM
|
7.0 | IC50 | 3 | Yes | |
XLCDJKIIBWOGQT
|
7.0 | IC50 | 3 | Yes | |
FXUWJFZELUGOAQ
|
7.0 | IC50 | 3 | Yes | |
GGYBWFRTPPVUAZ
|
6.9 | IC50 | 4 | Yes | |
LOTUNSOIIWVNBG
|
6.9 | Ki | 2 | — | |
XZAGAORJLXBQCC
|
6.9 | IC50 | 4 | Yes | |
JOTYZMGPCUSZKL
|
6.9 | IC50 | 2 | — | |
CADNLTAFOMUWRR
|
6.9 | IC50 | 3 | Yes | |
CDQQKPZINNWUDS
|
6.9 | IC50 | 2 | — | |
OKGOBXODUWTHAJ
|
6.9 | IC50 | 3 | Yes | |
QOWBVKQSFCSJAK
|
6.8 | IC50 | 5 | — | |
QTXVPJOTKLUYMQ
|
6.8 | IC50 | 5 | — | |
QQKFJAPYPOIWRW
|
6.8 | IC50 | 3 | Yes | |
VXPAAABROXRBQT
|
6.8 | IC50 | 3 | Yes | |
HOYBUULCSXDSPC
|
6.8 | IC50 | 3 | Yes | |
IIBLNMYMPDUKOQ
|
6.8 | Ki | 3 | Yes | |
SPGSQKKTHWOODB
|
6.8 | IC50 | 3 | Yes | |
XKPUKZQRNSFQLM
|
6.8 | IC50 | 3 | Yes | |
KAJHXHOIEARPHN
|
6.7 | IC50 | 2 | Yes | |
ODKWXUUQJAZOOR
|
6.7 | IC50 | 2 | — | |
QHTFXHUNNOAYME
|
6.7 | IC50 | 2 | — | |
MWMRJYLEVAWDDL
|
6.7 | IC50 | 7 | Yes | |
IDLHJNPBZBJSDO
|
6.7 | IC50 | 3 | Yes | |
ZFHJWQWVJPMAIW
|
6.7 | IC50 | 4 | Yes | |
YAYGKNVDBLFWFW
|
6.6 | IC50 | 6 | Yes | |
CNUCYIDHDPTDOD
|
6.6 | Ki | 5 | Yes | |
AFJYAUBLMRWZHB
|
6.5 | IC50 | 2 | — | |
KMMSPMPORWBMTE
|
6.5 | IC50 | 4 | Yes | |
NJCBPLQYZDLBCA
|
6.5 | IC50 | 3 | Yes | |
MITLEGOYVUMBJH
|
6.5 | IC50 | 3 | Yes | |
RINLHBFSMHCDCB
|
6.5 | IC50 | 3 | Yes | |
QWCJOBSHHHILCA
|
6.4 | IC50 | 3 | Yes |