Target Details
| UniProt AC | O14672 |
|---|---|
| Gene Symbol | ADAM10 |
| Protein Name | Disintegrin and metalloproteinase domain-containing protein 10 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21299 (ADAM10_Cys-rich) PF00200 (Disintegrin) PF13574 (Reprolysin_2) |
Summary
- Multi-target molecules 111
- Clinical molecules 78
- Avg pChEMBL 7.16
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (111)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GHVMTHKJUAOZJP
|
8.3 | IC50 | 2 | — | |
RFPBLNFCSNMAEW
|
8.3 | IC50 | 2 | — | |
ZKFYETVHOLUSNG
|
8.1 | IC50 | 7 | Yes | |
YDJAXPJDHWQNLF
|
8.1 | IC50 | 4 | Yes | |
FWILDXURZVZYSC
|
8.0 | IC50 | 3 | — | |
PDNKMRBXZXHUFT
|
8.0 | IC50 | 4 | Yes | |
JRYQAIVHIZIBOQ
|
8.0 | IC50 | 3 | Yes | |
VLUAXQQDRZDFOF
|
8.0 | IC50 | 3 | Yes | |
YLTJCMLZAIRVFF
|
8.0 | IC50 | 2 | — | |
FQUKTXLABCFONX
|
7.9 | IC50 | 3 | Yes | |
JGSJEYLQTZAQRG
|
7.9 | IC50 | 7 | Yes | |
GMXIFCSQVFGFBC
|
7.8 | IC50 | 3 | Yes | |
SPGSQKKTHWOODB
|
7.8 | IC50 | 4 | Yes | |
PWJXCFJUGNPSAZ
|
7.8 | IC50 | 2 | — | |
RTBFVYBTGAGBSP
|
7.8 | IC50 | 3 | Yes | |
VVHOXHYIVMZQIO
|
7.8 | IC50 | 2 | — | |
YYMXPNNILUETLE
|
7.7 | IC50 | 3 | Yes | |
JUKNHBAVDHQUJP
|
7.7 | IC50 | 3 | Yes | |
KRVYWSXTKLCPHD
|
7.7 | IC50 | 3 | Yes | |
CTRWITLGGIGPOB
|
7.7 | IC50 | 2 | — | |
KMMXFFDNBCQBEI
|
7.7 | IC50 | 3 | Yes | |
KSBCPHOBEZMZNM
|
7.7 | IC50 | 4 | Yes | |
ZABUEZYWKJKVJI
|
7.7 | IC50 | 2 | — | |
CKZHFOKQZRZCPF
|
7.7 | IC50 | 9 | Yes | |
FYZPCUXRTDXRBF
|
7.7 | IC50 | 6 | Yes | |
VVWOQMJGNBQWHG
|
7.6 | IC50 | 3 | Yes | |
ZCDHAHOTIYZFKF
|
7.6 | IC50 | 7 | Yes | |
WKQUYZQZMVHYFW
|
7.6 | IC50 | 2 | — | |
IDSXRTDVRWTZOK
|
7.6 | IC50 | 7 | Yes | |
MIUJFEWUCGLALV
|
7.6 | IC50 | 4 | Yes | |
GHVMTHKJUAOZJP
|
7.6 | IC50 | 6 | — | |
LIKQSFURRNSUMR
|
7.5 | Ki | 2 | — | |
AVCGYVHCLDMOAW
|
7.5 | IC50 | 3 | Yes | |
DAWQVDWNIUMYHC
|
7.5 | IC50 | 2 | Yes | |
FQSNZGGDFVIKEV
|
7.5 | IC50 | 4 | Yes | |
ZMPZOWIAKRPTEQ
|
7.5 | IC50 | 3 | Yes | |
MHXODSYUSQLZGR
|
7.5 | IC50 | 6 | Yes | |
SCOVLRMEIYKGOU
|
7.5 | IC50 | 6 | Yes | |
PFMDDCHUGSRIJN
|
7.5 | IC50 | 4 | Yes | |
YZXVQIOBIKCYRB
|
7.5 | IC50 | 2 | Yes | |
NITYDPDXAAFEIT
|
7.3 | IC50 | 20 | Yes | |
OCSMOTCMPXTDND
|
7.3 | IC50 | 14 | Yes | |
PEAOAVRAGQRJEO
|
7.3 | IC50 | 4 | Yes | |
ZOHXHAYMXURWLP
|
7.3 | IC50 | 3 | Yes | |
BTZCYRDTCBYYDO
|
7.3 | IC50 | 2 | — | |
JWVKYLLQNXGDRB
|
7.2 | IC50 | 5 | Yes | |
SPGSQKKTHWOODB
|
7.2 | IC50 | 3 | Yes | |
VPNMZNYQFRFELQ
|
7.2 | IC50 | 4 | Yes | |
YQLRSUQLXQKLGB
|
7.2 | IC50 | 2 | — | |
JLFCWOIZNQXZMP
|
7.2 | IC50 | 3 | Yes |