Target Details
UniProt ACO00591
Gene SymbolGABRP
Protein NameGamma-aminobutyric acid receptor subunit pi
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 325
  • Clinical molecules 0
  • Avg pChEMBL 7.41
Top Co-occurrence Targets
Active Molecules (325)
InChIKey pChEMBL Type Targets Clinical
VDAHGXKTABYDOQ 7.0 Ki 16
XJSZCKCJAMOVEP 7.0 IC50 16
OWUSBEXUSSJSDZ 7.0 IC50 16
KQTMWRZAVOUNCI 7.0 IC50 16
IIDOALWZHDFUQF 7.0 IC50 16
FQDQLHDSVITISC 7.0 IC50 16
YEFFWDGMWBFKHL 7.0 Ki 16
RMGFIVKKLZZKNY 7.0 IC50 16
XVRONCOEBFKZEW 7.0 IC50 16
NMMJOCVBNVTBNP 6.9 Ki 16
GQXSRHIFUJLCSW 6.9 Ki 16
JYXHNHBKWZQGLB 6.9 Ki 16
HWOWPGLTTSFLOQ 6.9 Ki 16
VFKHADGYGKHTDK 6.9 IC50 16
LHSWKUZVAZKLHJ 6.9 IC50 16
VFPUCBWBLOQFPU 6.9 IC50 16
YZBJLGYBBNTKKL 6.9 IC50 16
VHBFFQKBGNRLFZ 6.9 Ki 21
ACPUCHLYONVNTK 6.9 Ki 16
XYLGLGFZLQRDKD 6.9 Ki 16
BIHMYZHWJAFHBO 6.8 IC50 16
KOTFZRCPKVQWPP 6.8 Ki 16
XLKFCRQJPWBJNW 6.8 IC50 16
KTFRBKXLNKKPEA 6.8 IC50 16
DGWAMRKYNYINRJ 6.8 IC50 16
QQXJSYFEJVOQLZ 6.8 IC50 16
VGZQARXDBOOWBF 6.8 Ki 16
JTQDBIFZWJTIIQ 6.8 Ki 16
JXKAURVNHHPPND 6.8 IC50 16
RHARCGZTSJROQQ 6.8 Ki 16
RLKPTPBBRCFHEK 6.8 IC50 16
BXKSCEUJEPDZBI 6.8 Ki 16
STQWWORVIGBLOE 6.8 Ki 16
XAXZXMJZHNVJEQ 6.8 Ki 16
CGOOGLSJSVATGZ 6.8 Ki 16
FLHRNVLCKMTQAP 6.8 Ki 17
JQHJWKNJYLNAFL 6.8 IC50 16
XLKFCRQJPWBJNW 6.8 IC50 16
CGVJPQYHXQIFPE 6.7 Ki 16
PGTVWKLGGCQMBR 6.7 IC50 16
QKZNNAUSAVZXNE 6.7 Ki 16
HGPFVUUTSFNGNR 6.7 Ki 18
GMVMGIYPRPPNMB 6.7 Ki 16
ZRKQHHNVLRRZFQ 6.7 Ki 16
PTRPQDMPYNOBTR 6.7 IC50 16
DATCQVJMADOCRS 6.7 IC50 16
GXUSNZYZTBJMIT 6.7 Ki 16
SINAJPKUKOSXOT 6.7 IC50 16
WFRRJMYHDPXXFB 6.7 Ki 16
YWCLXVVWMQVKRF 6.7 IC50 16
2D structure