Target Details
| UniProt AC | O00444 |
|---|---|
| Gene Symbol | PLK4 |
| Protein Name | Serine/threonine-protein kinase PLK4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18190 (Plk4_PB1) PF18409 (Plk4_PB2) |
Summary
- Multi-target molecules 542
- Clinical molecules 39
- Avg pChEMBL 7.64
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (542)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KGXBCWANASZZQG
|
7.1 | IC50 | 5 | — | |
JAHXQCZCZURPTI
|
7.1 | IC50 | 34 | — | |
ANCOGLNFWMGEPC
|
7.1 | IC50 | 2 | — | |
LQVXSNNAFNGRAH
|
7.1 | Kd | 33 | Yes | |
JBZRAEUHDPMQSF
|
7.0 | IC50 | 34 | — | |
ZCCPLJOKGAACRT
|
7.0 | Kd | 599 | — | |
HCCIPHZGDVGCQS
|
7.0 | IC50 | 2 | — | |
QSTZYQDJSHNEIC
|
7.0 | IC50 | 2 | — | |
GIWIOFZXFSKQTE
|
7.0 | IC50 | 4 | — | |
JOOXLOJCABQBSG
|
7.0 | Kd | 139 | — | |
CNTCGRJDUJEUDG
|
7.0 | Ki | 37 | — | |
DFMCXVONDDGQIY
|
7.0 | Ki | 66 | — | |
GSXRCPJTNIGKSZ
|
7.0 | Ki | 43 | — | |
ITTRLTNMFYIYPA
|
7.0 | Kd | 17 | — | |
LGHBDVLAHHANMX
|
7.0 | Ki | 53 | — | |
SBFPHSVZEXSHTL
|
7.0 | Ki | 62 | — | |
DUBHPLWTLUVGNU
|
7.0 | IC50 | 5 | — | |
AWDORCFLUJZUQS
|
6.9 | Ki | 7 | — | |
KDKUVYLMPJIGKA
|
6.9 | Kd | 91 | Yes | |
TUBXJQSNTKADJB
|
6.9 | IC50 | 5 | — | |
CXBBWVXSZINRCS
|
6.9 | Ki | 41 | — | |
GWMATETWMAQOFL
|
6.9 | Ki | 36 | — | |
JZTOUVBEZONDKA
|
6.9 | Ki | 80 | — | |
MHCPAORAYMTGCZ
|
6.9 | Ki | 37 | — | |
NRZYTPAJGVTKIM
|
6.9 | Ki | 38 | — | |
QJIVDCJIPGAKQZ
|
6.9 | Ki | 25 | — | |
QONPPIZSNSSCSK
|
6.9 | Ki | 45 | Yes | |
XUGXUDSTKPTWNB
|
6.9 | Ki | 10 | — | |
ZVWRFVCNQOECJS
|
6.9 | Ki | 71 | — | |
BLQYVHBZHAISJM
|
6.9 | Kd | 21 | Yes | |
DUKJABPGWUISRC
|
6.9 | IC50 | 10 | — | |
FMRUHQLKCRUMNL
|
6.9 | IC50 | 4 | — | |
KTEIFNKAUNYNJU
|
6.8 | Ki | 48 | — | |
SHPFDGWALWEPGS
|
6.8 | Kd | 35 | — | |
DZSUJUOJJJCWGG
|
6.8 | Ki | 55 | Yes | |
AWDORCFLUJZUQS
|
6.8 | Ki | 22 | — | |
FQEODTMNWMDUMD
|
6.8 | Ki | 25 | — | |
GALVWTFFXPRMQM
|
6.8 | Ki | 20 | — | |
GLMWKEAUVZDGKE
|
6.8 | Ki | 23 | — | |
GQLWKGVBOIYMTN
|
6.8 | Ki | 35 | — | |
IFQICUARAXVEIQ
|
6.8 | Ki | 18 | — | |
LVECPYVAIBNSRV
|
6.8 | Ki | 33 | — | |
NLUPJKQOKWBWFC
|
6.8 | Ki | 69 | — | |
OLUKILHGKRVDCT
|
6.8 | Ki | 44 | Yes | |
PNKALLUVKOKYHZ
|
6.8 | Ki | 32 | — | |
SFPWNTQWFFNJIH
|
6.8 | Ki | 48 | — | |
ZGDSBEUMPIMXBM
|
6.8 | Ki | 42 | — | |
ZKHDDJKHTPLPOQ
|
6.8 | Ki | 62 | — | |
HXHAJRMTJXHJJZ
|
6.8 | Ki | 52 | Yes | |
CTNPALGJUAXMMC
|
6.7 | Kd | 151 | — |