Target Details
| UniProt AC | O00444 |
|---|---|
| Gene Symbol | PLK4 |
| Protein Name | Serine/threonine-protein kinase PLK4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18190 (Plk4_PB1) PF18409 (Plk4_PB2) |
Summary
- Multi-target molecules 542
- Clinical molecules 39
- Avg pChEMBL 7.64
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (542)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KNARVZUUCLIBGV
|
7.4 | Ki | 33 | — | |
UDFDIIVNIYWXDM
|
7.4 | Ki | 74 | — | |
WKEYMNLZBZKLOG
|
7.4 | Ki | 14 | — | |
XHORJSJFHVABEA
|
7.4 | Ki | 49 | — | |
XJSFDMGICAWQFS
|
7.4 | Ki | 60 | — | |
ZLHFILGSQDJULK
|
7.4 | Ki | 37 | Yes | |
WKDACQVEJIVHMZ
|
7.4 | Kd | 46 | — | |
CPKWRHVMDOSXKE
|
7.4 | IC50 | 5 | — | |
CQJVDJZHNQFAOH
|
7.3 | IC50 | 2 | — | |
DFZUUTZHVCYKTM
|
7.3 | IC50 | 2 | — | |
OOMBFNDWQIGHEK
|
7.3 | Kd | 22 | — | |
BIKYDWLMTPRSQL
|
7.3 | Ki | 50 | — | |
FAYAUAZLLLJJGH
|
7.3 | Ki | 36 | Yes | |
KKYPRNBBPBRJQX
|
7.3 | Ki | 40 | — | |
NFKMFNBKEOQNPZ
|
7.3 | Ki | 43 | — | |
NRGYZNJPCGRCLV
|
7.3 | Ki | 52 | — | |
TVLFEDKEAOXRCZ
|
7.3 | Ki | 22 | — | |
ULTZAKUJXNGGGZ
|
7.3 | IC50 | 2 | — | |
SLEWGGZPOQNVSU
|
7.3 | Kd | 22 | — | |
XZXHXSATPCNXJR
|
7.3 | Kd | 165 | Yes | |
IKVNNBYIDXRNMG
|
7.3 | IC50 | 3 | — | |
JRLOPMVTMMPZMV
|
7.2 | IC50 | 6 | — | |
KTEIFNKAUNYNJU
|
7.2 | Kd | 114 | — | |
ADLPKFFMGIJZIM
|
7.2 | Ki | 44 | — | |
AZTMYWWWILJAKW
|
7.2 | Ki | 16 | Yes | |
HKZKELVPGXJIMW
|
7.2 | Ki | 41 | — | |
LRZYYIZFBXFSJB
|
7.2 | Ki | 69 | — | |
NHFDRBXTEDBWCZ
|
7.2 | Ki | 41 | — | |
OWFLADWRSCINST
|
7.2 | Ki | 30 | — | |
PTVPBWWDGZSEAF
|
7.2 | Ki | 63 | — | |
RTDSHUGNRVXRHN
|
7.2 | Ki | 51 | — | |
VKBFHTIUXUCYRQ
|
7.2 | Ki | 66 | — | |
XBYVOPRDASFDMY
|
7.2 | Ki | 42 | — | |
TWURNGNKPCPSAH
|
7.2 | IC50 | 2 | — | |
BMGQWWVMWDBQGC
|
7.2 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
7.2 | Kd | 91 | Yes | |
MFAQYJIYDMLAIM
|
7.2 | Kd | 130 | Yes | |
MGGBYMDAPCCKCT
|
7.2 | Kd | 23 | — | |
KOZFSFOOLUUIGY
|
7.1 | Kd | 88 | Yes | |
NMIDELFSFNCISG
|
7.1 | IC50 | 2 | — | |
PXZRCYBRDGOXPD
|
7.1 | IC50 | 3 | — | |
CPPKXSQKLCJLNX
|
7.1 | IC50 | 2 | — | |
DBXGGXLBTWZXBB
|
7.1 | Ki | 39 | — | |
JAMDNXUAYUHJLJ
|
7.1 | Ki | 40 | — | |
MPFUDUPAOWHBRQ
|
7.1 | IC50 | 2 | — | |
MULNSLQVKKUPJN
|
7.1 | Ki | 41 | — | |
OWDRQHVEJIYVOI
|
7.1 | Ki | 47 | — | |
UGEJLCNSVIVALC
|
7.1 | Ki | 41 | — | |
ULHGAQSVFPOUDY
|
7.1 | Ki | 43 | — | |
ZGZVRPRSFXRGCF
|
7.1 | Ki | 76 | — |