Target Details
| UniProt AC | O00444 |
|---|---|
| Gene Symbol | PLK4 |
| Protein Name | Serine/threonine-protein kinase PLK4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18190 (Plk4_PB1) PF18409 (Plk4_PB2) |
Summary
- Multi-target molecules 542
- Clinical molecules 39
- Avg pChEMBL 7.64
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (542)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ODVQNAZETSWKTM
|
7.8 | IC50 | 2 | — | |
RBXYGQNZRVPDNB
|
7.8 | Ki | 34 | — | |
RITAVMQDGBJQJZ
|
7.8 | IC50 | 43 | — | |
ZCCJKVBTHCOISJ
|
7.8 | Ki | 46 | — | |
DJXMOVBYEXHLBK
|
7.8 | IC50 | 2 | — | |
IXAOAKWGJQGTSH
|
7.8 | IC50 | 3 | — | |
JEWLTBAFKJFWSC
|
7.7 | IC50 | 2 | — | |
CXQHYVUVSFXTMY
|
7.7 | Kd | 154 | — | |
IAKGNUWZPSPEKU
|
7.7 | Ki | 19 | — | |
KJLHICWSHQCTOG
|
7.7 | IC50 | 2 | — | |
LYNBNVBMAGDJRW
|
7.7 | Ki | 81 | — | |
MVJMMLFMPWITEJ
|
7.7 | Ki | 110 | — | |
OSVUGUHRKMMBSE
|
7.7 | Kd | 170 | — | |
RITAVMQDGBJQJZ
|
7.7 | Ki | 33 | — | |
LOLPPWBBNUVNQZ
|
7.7 | Kd | 97 | Yes | |
NKZIDRRJDMHQEU
|
7.7 | IC50 | 2 | — | |
YYLKKYCXAOBSRM
|
7.7 | Kd | 191 | — | |
AVAVKQHLKBUJPO
|
7.7 | IC50 | 3 | — | |
NAVCZBYGYNEESQ
|
7.7 | IC50 | 2 | — | |
UHXOAJSLKLIFLJ
|
7.7 | IC50 | 2 | — | |
JWODVWOSUKHGSK
|
7.6 | IC50 | 2 | — | |
AVDISIKMHVXATN
|
7.6 | IC50 | 2 | — | |
VYVQQIIOKNXZRD
|
7.6 | IC50 | 2 | — | |
XXIGPMYXABVGBW
|
7.6 | IC50 | 2 | — | |
BLQYVHBZHAISJM
|
7.6 | Ki | 54 | — | |
IOBVCHJTLVPPBR
|
7.6 | Ki | 39 | — | |
VYTKFXBQPJOMSD
|
7.6 | IC50 | 2 | — | |
XKZINYYXWJEYEL
|
7.6 | Ki | 37 | — | |
GFUZUEVAWXYASP
|
7.6 | IC50 | 3 | — | |
OEHGEOWDIWFUCT
|
7.6 | IC50 | 2 | — | |
LBVPYCHFUOFKSH
|
7.6 | IC50 | 2 | — | |
GPIAZIBOIDFMKV
|
7.6 | IC50 | 2 | — | |
NLPZXQSEMRVFPW
|
7.5 | IC50 | 2 | — | |
VMUFFHDFTBDUIP
|
7.5 | IC50 | 2 | — | |
CSCUXLKCEJASIE
|
7.5 | IC50 | 2 | — | |
GUBJNPWVIUFSTR
|
7.5 | Kd | 103 | — | |
RJZDECGDCKOHBV
|
7.5 | Ki | 70 | — | |
XOOAAYRIVATZNM
|
7.5 | Ki | 55 | — | |
YFNWWNRZJGMDBR
|
7.5 | Kd | 35 | — | |
WAVGXEMZTAFUCY
|
7.5 | IC50 | 2 | — | |
DKZYXHCYPUVGAF
|
7.5 | Kd | 112 | — | |
NXSJMRCTGYTSTK
|
7.5 | Kd | 200 | — | |
GTSAWXOXCVPESK
|
7.5 | IC50 | 2 | — | |
CIBNJPAPNFXEMP
|
7.5 | IC50 | 3 | — | |
KJZLFAOURNOQKC
|
7.5 | IC50 | 3 | — | |
AJZIGZOVWAFSBH
|
7.4 | IC50 | 2 | — | |
ZXCYXMDSRPHJRK
|
7.4 | IC50 | 2 | — | |
AOBLBPWPSKBHSI
|
7.4 | Ki | 55 | — | |
FQYLJBVSYHZWLT
|
7.4 | Ki | 35 | Yes | |
HAYYBYPASCDWEQ
|
7.4 | Ki | 47 | — |