Target Details
| UniProt AC | O00444 |
|---|---|
| Gene Symbol | PLK4 |
| Protein Name | Serine/threonine-protein kinase PLK4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18190 (Plk4_PB1) PF18409 (Plk4_PB2) |
Summary
- Multi-target molecules 542
- Clinical molecules 39
- Avg pChEMBL 7.64
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (542)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NRFMLFPXDKIQBF
|
8.5 | Kd | 8 | — | |
ALKJNCZNEOTEMP
|
8.5 | Kd | 55 | — | |
IICOWTOEYHWWOH
|
8.5 | IC50 | 3 | — | |
MHWMTNNCBDPEDS
|
8.5 | IC50 | 2 | — | |
SCIOAYVRXBCGMK
|
8.5 | IC50 | 2 | — | |
OWRXHGAFWZFFCW
|
8.5 | Ki | 113 | — | |
LDGOZDNOQAZRQV
|
8.5 | IC50 | 2 | — | |
CBRMHVZZHXKJJW
|
8.5 | IC50 | 2 | — | |
FQSHTSWWNWIELG
|
8.5 | IC50 | 3 | — | |
MOVPUGMNBIXRIN
|
8.5 | IC50 | 2 | — | |
VDOFAJCHUPIPJF
|
8.5 | IC50 | 2 | — | |
UZFYLZWGFGEELR
|
8.5 | IC50 | 3 | — | |
VWVYILCFSYNJHF
|
8.5 | Ki | 49 | — | |
SEJGTFPOEJWEGG
|
8.5 | Kd | 149 | — | |
LYTYIKFSJLZITL
|
8.4 | IC50 | 2 | — | |
BUMGKNPRCXMAGM
|
8.4 | IC50 | 6 | — | |
CZFUYZPXZGGWKC
|
8.4 | IC50 | 7 | — | |
PYWVRRARNRCHNK
|
8.4 | IC50 | 2 | — | |
FUWXNWLFYOEPCL
|
8.4 | IC50 | 2 | — | |
GSMALWRBDKEIGI
|
8.4 | IC50 | 2 | — | |
HYQVDRMLTQMPMN
|
8.4 | IC50 | 2 | — | |
QKHVOBMZVQSXAS
|
8.4 | IC50 | 2 | — | |
GYMQBVYIGPAFNJ
|
8.4 | IC50 | 2 | — | |
HCLJFCCORISDCX
|
8.4 | IC50 | 5 | — | |
HTHISIOYCCJIBY
|
8.4 | IC50 | 2 | — | |
UYJNQQDJUOUFQJ
|
8.4 | Ki | 68 | — | |
JJQRFOFBCUENFJ
|
8.4 | IC50 | 2 | — | |
VTCVDQBVMWVWLM
|
8.4 | IC50 | 2 | — | |
UZTAKXKQQVMUNQ
|
8.3 | IC50 | 3 | — | |
NNCYMIKCSDIHJR
|
8.3 | IC50 | 3 | — | |
AHXHWEURVLCQAX
|
8.3 | IC50 | 2 | — | |
VOJAEHGONMEHQB
|
8.3 | IC50 | 2 | — | |
DQTLTCIEAKFGBZ
|
8.3 | IC50 | 3 | — | |
VXWLORZXKCHFJR
|
8.3 | IC50 | 2 | — | |
GBIUARDTAPJECU
|
8.3 | IC50 | 2 | — | |
XKFTZKGMDDZMJI
|
8.3 | Kd | 64 | Yes | |
XSXNOQJYDZWMGX
|
8.3 | IC50 | 2 | — | |
DEQUZSQDCDHROJ
|
8.3 | IC50 | 2 | — | |
XCDJZSMEKBJHEE
|
8.2 | IC50 | 2 | — | |
SBEXUUCHJQBRNW
|
8.2 | IC50 | 2 | — | |
UYYCHKFCCDPBMQ
|
8.2 | IC50 | 3 | — | |
XVTGWJWSWNCTFK
|
8.2 | IC50 | 3 | — | |
IWDQHFKKTHSUKI
|
8.2 | IC50 | 2 | — | |
LDGOZDNOQAZRQV
|
8.2 | IC50 | 2 | — | |
IXIQSDVVXYFVAG
|
8.2 | IC50 | 2 | — | |
ALZQFLLQPOLVEW
|
8.2 | IC50 | 2 | — | |
FQIKRDSTMHHCGU
|
8.2 | IC50 | 3 | — | |
LICZLVVAGKBEKQ
|
8.2 | IC50 | 3 | — | |
LIUOIZMHHPJCCK
|
8.2 | IC50 | 2 | — | |
PDOXJVQIOMGRBV
|
8.2 | IC50 | 2 | — |