Target Details
| UniProt AC | O00444 |
|---|---|
| Gene Symbol | PLK4 |
| Protein Name | Serine/threonine-protein kinase PLK4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18190 (Plk4_PB1) PF18409 (Plk4_PB2) |
Summary
- Multi-target molecules 542
- Clinical molecules 39
- Avg pChEMBL 7.64
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (542)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GJFMMVDSDLIPNN
|
8.8 | IC50 | 2 | — | |
RBNRSVPXZPBXCD
|
8.8 | IC50 | 5 | — | |
AMKGWZMBMZFCTO
|
8.7 | IC50 | 3 | — | |
JHIXLFUYHWBARZ
|
8.7 | IC50 | 2 | — | |
UEMHNDHVZSSWDQ
|
8.7 | IC50 | 2 | — | |
GLQBCBXEXHJHCZ
|
8.7 | IC50 | 2 | — | |
HELHZUKLOPVPHW
|
8.7 | IC50 | 3 | — | |
VVFYYEUTPUGPNR
|
8.7 | IC50 | 2 | — | |
WIYXOIDCQNFVET
|
8.7 | IC50 | 3 | — | |
WUTLVPJTLNYGRZ
|
8.7 | IC50 | 2 | — | |
CFIBXVQLBVNOHW
|
8.7 | Ki | 64 | — | |
FYDMEKZWCPHGNB
|
8.7 | IC50 | 2 | — | |
MEOINRRPIPRMSC
|
8.7 | IC50 | 2 | — | |
TZKMWKXQVXWVFE
|
8.7 | IC50 | 2 | — | |
ZWVVQRZMRVRZFD
|
8.7 | IC50 | 2 | — | |
FOJFMSKCYTZGMD
|
8.7 | IC50 | 3 | — | |
MAUAORFSSOOYOT
|
8.7 | IC50 | 2 | — | |
BSFSQSWHBCBLLD
|
8.7 | IC50 | 2 | — | |
BXCLMWKUQGBIJK
|
8.7 | IC50 | 2 | — | |
FDFNBHWHWWYCHN
|
8.7 | IC50 | 3 | — | |
RMGQWXVHWUUVLJ
|
8.7 | IC50 | 4 | — | |
AAEYSRYWDWVNOK
|
8.7 | IC50 | 2 | — | |
BNCUORANSSPIJN
|
8.7 | IC50 | 2 | — | |
LUPFUUDPZIMLMJ
|
8.7 | IC50 | 2 | — | |
JOCNOQUWDPPPRY
|
8.6 | IC50 | 2 | — | |
SXAOLYUXAFWLCI
|
8.6 | IC50 | 4 | — | |
UIJBTFOXBSSWCE
|
8.6 | IC50 | 2 | — | |
COYIMHAMNHOPTJ
|
8.6 | IC50 | 3 | — | |
MLSFACRPOXXXGI
|
8.6 | IC50 | 2 | — | |
OFJINLPIXOGONH
|
8.6 | IC50 | 2 | — | |
YCZYGQPCRPOGLT
|
8.6 | IC50 | 3 | — | |
ZRBJCFDMMPLPCO
|
8.6 | IC50 | 2 | — | |
GHVNNCGXWGZXJH
|
8.6 | IC50 | 4 | — | |
TVRYEYSLCUPRPL
|
8.6 | IC50 | 5 | — | |
QRDCBCOPUDYBCB
|
8.6 | IC50 | 4 | — | |
YSAUMHGSYAMXPK
|
8.6 | IC50 | 2 | — | |
HFEPCQCRRRINGD
|
8.6 | IC50 | 2 | — | |
JCDAVUJUCMYZTJ
|
8.6 | IC50 | 2 | — | |
WVGYXYZYFSSTFT
|
8.6 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
8.6 | Kd | 408 | — | |
JILOKERUAWMFHD
|
8.6 | IC50 | 3 | — | |
MMUWRPSFAYHCTP
|
8.6 | IC50 | 3 | — | |
WWFYNSPZDZAAER
|
8.6 | IC50 | 2 | — | |
AJWHDYZLFAUJLF
|
8.6 | IC50 | 2 | — | |
DMWCSOYJGHLVEB
|
8.6 | IC50 | 2 | — | |
HHJSKDRCUMVWKF
|
8.6 | IC50 | 7 | — | |
RKFHHTFCUQMIGM
|
8.6 | IC50 | 3 | — | |
UDFJBAMCRJJGMV
|
8.6 | IC50 | 2 | — | |
DADASRPKWOGKCU
|
8.6 | IC50 | 9 | — | |
MPUKOARMEBDIDZ
|
8.5 | IC50 | 2 | — |