Target Details
| UniProt AC | O00444 |
|---|---|
| Gene Symbol | PLK4 |
| Protein Name | Serine/threonine-protein kinase PLK4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18190 (Plk4_PB1) PF18409 (Plk4_PB2) |
Summary
- Multi-target molecules 542
- Clinical molecules 39
- Avg pChEMBL 7.64
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (542)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MVKSHUDBXVAUPP
|
9.0 | IC50 | 2 | — | |
QYRNNGHSHFUOFR
|
9.0 | IC50 | 3 | — | |
NUALOIMAZAHWKR
|
9.0 | IC50 | 2 | — | |
NZBZBQUHFXSFOR
|
9.0 | IC50 | 4 | — | |
VZTSXPRAPGCSCR
|
9.0 | IC50 | 2 | — | |
CGFXXKQAUTXPSO
|
8.9 | IC50 | 2 | — | |
OHDDAHALDZFALJ
|
8.9 | IC50 | 3 | — | |
QACPKRRQDDUBDE
|
8.9 | IC50 | 3 | — | |
YLDZSOOIPBFXEN
|
8.9 | IC50 | 3 | — | |
NTNIBJDMRRLYOK
|
8.9 | IC50 | 2 | — | |
NHXVTGGWJAZMKU
|
8.9 | IC50 | 2 | — | |
OMFRMSODXLGAQT
|
8.9 | IC50 | 3 | — | |
PRDPUQGHWRZOIL
|
8.9 | IC50 | 3 | — | |
VIJMQSQDODLIHT
|
8.9 | IC50 | 3 | — | |
CRIUUFBOLAJGNR
|
8.9 | IC50 | 3 | — | |
FPWMHTSISQKIJN
|
8.9 | IC50 | 2 | — | |
IVVSNTYYOLGITN
|
8.9 | IC50 | 2 | — | |
ZDXVFTIWQLMEIZ
|
8.9 | IC50 | 3 | — | |
DWBNOASTWMOBSP
|
8.9 | IC50 | 2 | — | |
JZIZUMLXHJPWJH
|
8.9 | IC50 | 2 | — | |
XMHCFCMVNKTYOH
|
8.9 | IC50 | 2 | — | |
ASHFSDTVSQCVQC
|
8.9 | IC50 | 2 | — | |
HOZCGFJBIZZKTL
|
8.9 | IC50 | 2 | — | |
CMLSWGVOCIGIAK
|
8.9 | IC50 | 2 | — | |
GWTSGLRTAKOPSF
|
8.9 | IC50 | 3 | — | |
PIHRITDRJRTFQR
|
8.9 | IC50 | 2 | — | |
USYYTOCVNAELEK
|
8.9 | IC50 | 3 | — | |
VSDZCJADMNPBKB
|
8.9 | IC50 | 3 | — | |
YNXZLNOLQBAZNQ
|
8.9 | IC50 | 3 | — | |
CKCGBVCGRTYHGB
|
8.9 | IC50 | 2 | — | |
FJKSYFWQWKRPJT
|
8.8 | IC50 | 2 | — | |
FQWPBCFJZAKNEQ
|
8.8 | IC50 | 4 | — | |
LLWIMNNGCHBSEF
|
8.8 | IC50 | 2 | — | |
SPVMVDXYFVXTKJ
|
8.8 | IC50 | 2 | — | |
HNFIGFQBTMODAW
|
8.8 | IC50 | 2 | — | |
HQCQFKQGMPBYGP
|
8.8 | IC50 | 4 | — | |
MRRJIJBPTGTPLV
|
8.8 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
8.8 | Kd | 289 | Yes | |
JXPRLYUMECVOOZ
|
8.8 | IC50 | 2 | — | |
YGKBBMAZIAXASO
|
8.8 | IC50 | 3 | — | |
ZVIBNYVMRHMJFS
|
8.8 | IC50 | 3 | — | |
DTPIGHJZEZDEAO
|
8.8 | IC50 | 3 | — | |
GBUDRABUNBYJKG
|
8.8 | IC50 | 7 | — | |
KMNQWCTYNHJINU
|
8.8 | IC50 | 2 | — | |
USCOCXHLSIVHKU
|
8.8 | IC50 | 3 | — | |
YTALSCBTOISJNF
|
8.8 | IC50 | 2 | — | |
DBLHAVCJDSOAAZ
|
8.8 | IC50 | 2 | — | |
UOUWRLIIMOCVBC
|
8.8 | IC50 | 3 | — | |
NGQVGKKCRFIRQR
|
8.8 | IC50 | 3 | — | |
DZSFRHLIEUXICV
|
8.8 | IC50 | 2 | — |