Target Details
| UniProt AC | O00444 |
|---|---|
| Gene Symbol | PLK4 |
| Protein Name | Serine/threonine-protein kinase PLK4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18190 (Plk4_PB1) PF18409 (Plk4_PB2) |
Summary
- Multi-target molecules 542
- Clinical molecules 39
- Avg pChEMBL 7.64
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (542)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MZDKLVOWGIOKTN
|
6.2 | Ki | 80 | — | |
RPGBQFNDFPEOON
|
6.2 | Ki | 22 | — | |
WVFWTUJEHMVUBG
|
6.2 | Ki | 25 | — | |
AYCPARAPKDAOEN
|
6.2 | Kd | 73 | — | |
JRLOPMVTMMPZMV
|
6.2 | IC50 | 4 | — | |
VRWFLNVDDMVVDA
|
6.2 | IC50 | 7 | — | |
HJVFTUSVRMGBLM
|
6.2 | IC50 | 7 | — | |
IAYGCINLNONXHY
|
6.1 | Kd | 50 | — | |
KRIUNPBAQZGFQA
|
6.1 | Kd | 76 | — | |
AUDNGNGLLRZLDR
|
6.1 | Ki | 33 | — | |
DKXHSOUZPMHNIZ
|
6.1 | Ki | 51 | Yes | |
FPQHXFMYXQZPSV
|
6.1 | Ki | 23 | — | |
JSDGKSMNPHJDFK
|
6.1 | Ki | 35 | — | |
KTRGYJLQTZDGPX
|
6.1 | Ki | 9 | — | |
NKGLJTITEFZKAN
|
6.1 | Ki | 35 | — | |
QAJPIJHWTGPUNZ
|
6.1 | Ki | 37 | — | |
SHENEEFOURUIBP
|
6.1 | Ki | 29 | — | |
UPITUWGOTMBQLX
|
6.1 | Ki | 13 | — | |
XJJYJNMNYDNXNO
|
6.1 | Ki | 23 | — | |
XYZNKCSDQRKAFR
|
6.1 | Ki | 53 | — | |
ZZSBPGIGIUFJRA
|
6.1 | Kd | 46 | — | |
ZVPDNRVYHLRXLX
|
6.0 | Ki | 35 | Yes | |
BSFNGHCTZDCQBF
|
6.0 | Ki | 3 | — | |
AWJPVXSHMIELNJ
|
6.0 | Ki | 23 | — | |
CZGMEOAMQWAJOY
|
6.0 | IC50 | 15 | Yes | |
FDBPGAHVEGEARY
|
6.0 | Ki | 19 | — | |
GMYYMEOGFRKSFS
|
6.0 | Ki | 29 | — | |
IJVDETPCUCZHTR
|
6.0 | Ki | 12 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JCFJQIHDZHHMQT
|
6.0 | Ki | 42 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KNACLJBHKVSTDL
|
6.0 | Ki | 40 | — | |
KYACBMRLQMEIAI
|
6.0 | Ki | 30 | — | |
LKUJDAHYLPICSE
|
6.0 | Ki | 24 | — | |
LSFLAQVDISHMNB
|
6.0 | Ki | 13 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MIYRKQLKDQNUKZ
|
6.0 | Ki | 23 | — | |
PAIFYAZSILXLBO
|
6.0 | Ki | 26 | — | |
QNUKRWAIZMBVCU
|
6.0 | Ki | 46 | — | |
VBUWAJWPXASNGM
|
6.0 | Ki | 9 | — | |
VQPBIJGXSXEOCU
|
6.0 | Ki | 24 | — | |
ZCAOFAAOUBUUBJ
|
6.0 | Ki | 9 | — |