Target Details
| UniProt AC | O00444 |
|---|---|
| Gene Symbol | PLK4 |
| Protein Name | Serine/threonine-protein kinase PLK4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18190 (Plk4_PB1) PF18409 (Plk4_PB2) |
Summary
- Multi-target molecules 542
- Clinical molecules 39
- Avg pChEMBL 7.64
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (542)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JPOSFPUHBHRUAX
|
6.4 | IC50 | 40 | Yes | |
BTHLNBWTKKAULX
|
6.4 | Ki | 16 | — | |
DZIPQNPWTUXXSJ
|
6.4 | Ki | 18 | — | |
IUEBPIPDFMCSTP
|
6.4 | Ki | 29 | — | |
MFMXAWQGPQXDRJ
|
6.4 | Ki | 27 | — | |
OTVCFDOYUHREFJ
|
6.4 | Ki | 26 | — | |
QQUXFYAWXPMDOE
|
6.4 | Ki | 31 | — | |
RXVOXSGTUROJOL
|
6.4 | Ki | 11 | — | |
ULVWJFBHQIXEPE
|
6.4 | Ki | 10 | — | |
WICLISNBDMGFST
|
6.4 | Ki | 10 | — | |
WKWARMGSTJGPIX
|
6.4 | Ki | 3 | — | |
WUWDLXZGHZSWQZ
|
6.4 | Ki | 41 | — | |
ZMNWFTYYYCSSTF
|
6.4 | Ki | 18 | — | |
HGVSVCAZEMPVJS
|
6.4 | IC50 | 2 | — | |
HHFBDROWDBDFBR
|
6.4 | Kd | 40 | Yes | |
OYONTEXKYJZFHA
|
6.4 | Kd | 69 | Yes | |
PXSLUZICFBACPN
|
6.4 | IC50 | 2 | — | |
GWJHMRBQEUHFOC
|
6.4 | Ki | 3 | — | |
BWMYPJVJYVLPIC
|
6.3 | IC50 | 2 | — | |
ZULFKUINRYIZQT
|
6.3 | IC50 | 2 | — | |
AYJBHLUSGLQYDG
|
6.3 | Ki | 16 | — | |
DLWMVUDMPMKGEE
|
6.3 | Ki | 24 | — | |
FMPKTXNCNJCHCC
|
6.3 | Ki | 25 | — | |
FXQWJULRETZHHW
|
6.3 | Ki | 14 | — | |
GHMRUNOHAHJNNA
|
6.3 | Ki | 29 | — | |
ISVHLTLEHRZKJC
|
6.3 | Ki | 19 | — | |
JMHQUQCLIVNTHT
|
6.3 | Ki | 24 | — | |
MADCXGNPDBWPLM
|
6.3 | Ki | 25 | — | |
PEXKNSGOEOREKM
|
6.3 | Ki | 13 | — | |
PUPCRRRSBUYJAD
|
6.3 | Ki | 44 | Yes | |
RKUKAACYUCUJEE
|
6.3 | Ki | 58 | — | |
RWEHAHIEUDLKGT
|
6.3 | Ki | 33 | — | |
SPMHGQZFMNZCBV
|
6.3 | Ki | 30 | Yes | |
UTFXYGYVDDLJER
|
6.3 | Ki | 36 | — | |
WFTZMAAMCVPJJT
|
6.3 | Ki | 26 | — | |
ZLVOTRRGLSDLPF
|
6.3 | Ki | 36 | — | |
UKSUTRFTRYQMRC
|
6.3 | IC50 | 2 | — | |
BFSMGDJOXZAERB
|
6.3 | Kd | 33 | — | |
NZBZBQUHFXSFOR
|
6.3 | IC50 | 2 | — | |
UKGMAACIEPMUPX
|
6.3 | IC50 | 2 | — | |
UKGMAACIEPMUPX
|
6.3 | IC50 | 2 | — | |
YEZQDIPIXKWLNY
|
6.3 | IC50 | 2 | — | |
YEZQDIPIXKWLNY
|
6.3 | IC50 | 2 | — | |
GKDRMWXFWHEQQT
|
6.2 | Kd | 7 | — | |
QTBWCSQGBMPECM
|
6.2 | Kd | 21 | Yes | |
UHTHHESEBZOYNR
|
6.2 | Kd | 66 | Yes | |
GWJHMRBQEUHFOC
|
6.2 | Ki | 42 | — | |
HCNIBOQWDVOZKF
|
6.2 | Ki | 26 | — | |
LRLDYTTWQIFWBD
|
6.2 | Ki | 25 | — | |
MPVGZUGXCQEXTM
|
6.2 | Ki | 61 | Yes |