Target Details
| UniProt AC | O00444 |
|---|---|
| Gene Symbol | PLK4 |
| Protein Name | Serine/threonine-protein kinase PLK4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18190 (Plk4_PB1) PF18409 (Plk4_PB2) |
Summary
- Multi-target molecules 542
- Clinical molecules 39
- Avg pChEMBL 7.64
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (542)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WJHAMZUWDONFQH
|
10.0 | IC50 | 2 | — | |
JWPYZYBMSBDDCD
|
9.7 | IC50 | 2 | — | |
IYHJCLOZCBCODN
|
9.5 | IC50 | 2 | — | |
WNBOTPDRPIQGEY
|
9.5 | IC50 | 2 | — | |
XRPNCCIJNVBSFF
|
9.5 | IC50 | 2 | — | |
BXRQHDUUZXKTBX
|
9.5 | IC50 | 2 | — | |
CFVRISSXNGRSCL
|
9.4 | IC50 | 3 | — | |
OQYLKJLEFFUOSP
|
9.4 | IC50 | 3 | — | |
CNDHNCBFTRUZMZ
|
9.4 | IC50 | 2 | — | |
TVLISAFENSCERO
|
9.4 | IC50 | 2 | — | |
CHTYRUHQWURFTA
|
9.3 | IC50 | 3 | — | |
IYBUABKADRJAPB
|
9.2 | IC50 | 2 | — | |
PQNWGLHBIINSDV
|
9.2 | IC50 | 2 | — | |
DKVKUPRCFKTRIY
|
9.2 | IC50 | 7 | — | |
SRKLAYWRZKLNHC
|
9.2 | IC50 | 3 | — | |
TYJOLBATVWRDJW
|
9.2 | IC50 | 3 | — | |
RXKUYZFBEMBYSF
|
9.2 | IC50 | 2 | — | |
FQPRRMPEEHYYNP
|
9.2 | IC50 | 2 | — | |
HPYJNDCKRXOAKV
|
9.2 | IC50 | 2 | — | |
KHDTZPRXPIQIDD
|
9.2 | IC50 | 3 | — | |
HWDCMQBNOROFEQ
|
9.1 | IC50 | 2 | — | |
ZAYNEDGQOVESHF
|
9.1 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
9.1 | Kd | 213 | — | |
NEYBSPWSNSHKHW
|
9.1 | IC50 | 3 | — | |
CTKWGPSDOQLVKK
|
9.1 | IC50 | 2 | — | |
NYPQIYNAJRTAPS
|
9.1 | IC50 | 3 | — | |
HUKDVVBUBJTWCJ
|
9.1 | IC50 | 2 | — | |
RZBCOYUBQNCKGM
|
9.1 | IC50 | 3 | — | |
XTOHRNRFRAUJKC
|
9.1 | IC50 | 3 | — | |
MBNSFOGJHWUIOY
|
9.1 | IC50 | 2 | — | |
OJEKLDYMEMWETM
|
9.1 | IC50 | 2 | — | |
OZGUGQSGXNMCNT
|
9.1 | IC50 | 3 | — | |
QCHJTTRZNFGGKY
|
9.1 | IC50 | 2 | — | |
CODJRIKNYSCBSA
|
9.1 | IC50 | 3 | — | |
HZDOHYKYGNRPGO
|
9.1 | IC50 | 2 | — | |
QQWUGDVOUVUTOY
|
9.0 | Kd | 231 | Yes | |
ZSMPGSBOZTVRAJ
|
9.0 | IC50 | 3 | — | |
HTLXWQIMRWWAEB
|
9.0 | IC50 | 3 | — | |
RYEJQIGGOAKPKK
|
9.0 | IC50 | 3 | — | |
XIFWZYQJCXOJDM
|
9.0 | IC50 | 3 | — | |
GSYZCTCPLRSRGI
|
9.0 | IC50 | 2 | — | |
VHIUYJBYHQFWHD
|
9.0 | IC50 | 2 | — | |
AEINMBOZWWDMIV
|
9.0 | IC50 | 3 | — | |
CNMLMSRMIXOQJZ
|
9.0 | IC50 | 2 | — | |
DVCNPIFFEMVJNY
|
9.0 | IC50 | 3 | — | |
JAHZZERYOWPURL
|
9.0 | IC50 | 3 | — | |
PJIONPDTUIXVCT
|
9.0 | IC50 | 2 | — | |
ZNXHSLJBVPFPJV
|
9.0 | IC50 | 2 | — | |
JBOORGPMLIAKTP
|
9.0 | IC50 | 3 | — | |
MMCKCGTUACUYFW
|
9.0 | IC50 | 3 | — |