Target Details
UniProt ACO00443
Gene SymbolPIK3C2A
Protein NamePhosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit alpha
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00168 (C2) PF00454 (PI3_PI4_kinase) PF00792 (PI3K_C2) PF00794 (PI3K_rbd) PF00613 (PI3Ka) PF00787 (PX)
Summary
  • Multi-target molecules 128
  • Clinical molecules 0
  • Avg pChEMBL 7.53
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (128)
InChIKey pChEMBL Type Targets Clinical
OJWASAGOPPOBGC 9.2 IC50 2
HLTLYKPFSSMNIF 9.2 IC50 6
CQXNKRDLKVOXKL 9.2 IC50 3
PVSWNNSQKWFCQR 9.1 IC50 3
RDOPNBUYMXCSHN 9.1 IC50 2
CPUXOJVJEJZOSP 9.1 IC50 6
JCRXQCMCFXOERV 9.1 IC50 2
NMZOQFREGVBPSH 9.1 IC50 6
FEHPMLVVSQNYOF 9.1 IC50 7
JWVKJIWDNLLIHI 9.1 IC50 2
OEZASBKKYFBCDF 9.1 IC50 2
DVLVYFPEVHXTKT 9.1 IC50 6
ORLRMKPNSOWEHM 9.1 IC50 2
YLPQMLSKPUQHLB 9.1 IC50 6
QYMOZGDUAHTCOX 9.1 IC50 3
DFNYCHSSWGMVBA 9.0 IC50 3
YLPQMLSKPUQHLB 9.0 IC50 2
LHWJYPWCWCUOCY 9.0 IC50 3
RGXYXEURNXNTPI 9.0 IC50 2
UBTCFPBWLDOPTP 9.0 IC50 2
VOAMFTLRNNKOOY 9.0 IC50 3
WGDAYSZXELMOHH 9.0 IC50 2
CJBQWRITBDWUOS 9.0 IC50 2
ICBJQGXKICJHEP 9.0 IC50 2
IEDGFXCUFJCEAP 9.0 IC50 6
KYQCUZUJBXRUPX 9.0 IC50 2
LCKPXRGDNVKPOQ 9.0 IC50 2
LCMMFSOTAUQSFR 8.9 IC50 2
CBAOPIOAFUZMKL 8.9 IC50 2
GWPDIUMFLITIDY 8.9 IC50 2
SMNLEJPURJQOPX 8.8 IC50 3
YHSZNUBPVWCMDZ 8.8 IC50 2
IGXAFEIHWNLFBZ 8.8 IC50 3
LKTSHGKACAJSQF 8.8 IC50 3
MIIMBOHCWWMAIP 8.8 IC50 2
DVLVYFPEVHXTKT 8.7 IC50 2
UYOIRNOXDKRDHY 8.7 IC50 3
NAUZHEXCXBVBFU 8.7 IC50 2
TXSXEPQFXLQJNW 8.7 IC50 3
ATWVCAADDAUCNW 8.6 IC50 2
CWSKWYKUUUZDCL 8.6 IC50 2
RGSJELCNZVZCLI 8.6 IC50 2
SSQLNSGGUMJLAL 8.6 IC50 2
JZUROTPIGWBWRG 8.6 IC50 3
BEGSHQOQJPHHLL 8.6 IC50 3
UZVHGBFQKRNLCL 8.6 IC50 2
DBTUXAQQDZKWMP 8.4 IC50 2
PQWNEGGMCKZRSX 8.4 IC50 2
WCFYEDNZSHMOBJ 8.3 IC50 2
QNWUWGJORUNQBH 8.3 IC50 2
2D structure