Target Details
| UniProt AC | O00311 |
|---|---|
| Gene Symbol | CDC7 |
| Protein Name | Cell division cycle 7-related protein kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 484
- Clinical molecules 9
- Avg pChEMBL 7.69
KEGG Pathways (1)
Active Molecules (484)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LKUJDAHYLPICSE
|
6.2 | Ki | 24 | — | |
PCQMERRARZKTPW
|
6.2 | Ki | 68 | — | |
WHVFDYQCAMPLMS
|
6.2 | Ki | 20 | Yes | |
XBDWKVLCDCUNHH
|
6.2 | Ki | 18 | — | |
ZPVLRSVLOWVDJC
|
6.2 | Ki | 14 | — | |
ZVWRFVCNQOECJS
|
6.2 | Ki | 71 | — | |
MIYRKQLKDQNUKZ
|
6.2 | Ki | 23 | — | |
SAUBSLDUTDQGFT
|
6.2 | IC50 | 2 | — | |
ANMBSHUMLDUSAX
|
6.2 | IC50 | 4 | — | |
TXACPRMNHKOVDZ
|
6.2 | IC50 | 2 | — | |
LKQNORXYBMFYCG
|
6.2 | IC50 | 4 | — | |
ALCAFIIEVJETRN
|
6.1 | IC50 | 4 | — | |
WOYFMTIGVCKOTG
|
6.1 | IC50 | 2 | — | |
YXGFHFBKXWLFAZ
|
6.1 | IC50 | 4 | — | |
GUMBHNMWKMFKRT
|
6.1 | Ki | 23 | — | |
IUEBPIPDFMCSTP
|
6.1 | Ki | 29 | — | |
JCFJQIHDZHHMQT
|
6.1 | Ki | 42 | — | |
MWKSRKSEWLRPBL
|
6.1 | Kd | 1075 | — | |
SPOBBSBKXJKGBG
|
6.1 | Ki | 16 | — | |
VNGYQBMDQMDALH
|
6.1 | Ki | 25 | — | |
ZQVQTUFEKLITNT
|
6.1 | Ki | 10 | — | |
DRVZBNFJABEKEJ
|
6.1 | IC50 | 2 | — | |
BIVQAKMJEHVJCF
|
6.0 | IC50 | 2 | — | |
KOEWWBBSRQMABA
|
6.0 | Ki | 3 | — | |
FGNTZMWOEYXGLV
|
6.0 | IC50 | 2 | — | |
BFXKKVCGVIOJBH
|
6.0 | IC50 | 2 | — | |
IJVDETPCUCZHTR
|
6.0 | Ki | 12 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KRIUNPBAQZGFQA
|
6.0 | Ki | 76 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
ORMANVRRAHMNDI
|
6.0 | Ki | 2 | — | |
RFVBRKXQYUDGIO
|
6.0 | Ki | 23 | — | |
WYLVFMBGPRCDQF
|
6.0 | Ki | 14 | — |