Target Details
| UniProt AC | O00257 |
|---|---|
| Gene Symbol | CBX4 |
| Protein Name | E3 SUMO-protein ligase CBX4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17218 (CBX7_C) PF00385 (Chromo) |
Summary
- Multi-target molecules 23
- Clinical molecules 0
- Avg pChEMBL 6.66
KEGG Pathways (1)
Active Molecules (23)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UKWNWTBRKZUHGX
|
7.6 | Kd | 5 | — | |
ITTGNAWNEDCTNG
|
7.2 | IC50 | 3 | — | |
VWQADHAJYDYFRH
|
7.1 | IC50 | 3 | — | |
WKPAARGLUVBIGB
|
7.1 | IC50 | 4 | — | |
SQWGTAUPVFPVAQ
|
7.0 | Kd | 2 | — | |
UMRRDXVUROEIKJ
|
7.0 | Kd | 5 | — | |
VLYHVKRJXDXUFJ
|
7.0 | IC50 | 3 | — | |
QEMFCTCDHJQLGF
|
6.8 | IC50 | 3 | — | |
ROYGCJFTRGCLIU
|
6.8 | IC50 | 3 | — | |
IQFBELGVMQWYDI
|
6.8 | IC50 | 3 | — | |
SOGNIQLFQOQYGJ
|
6.7 | IC50 | 3 | — | |
AEXWIZIRHCUOMT
|
6.7 | IC50 | 3 | — | |
LGOXKBJUNDKRRI
|
6.7 | Kd | 5 | — | |
PBCHJNMDDNVDMG
|
6.6 | IC50 | 3 | — | |
RVSBUVWESBGOMR
|
6.5 | Kd | 2 | — | |
YKZYTGMDKIVZKB
|
6.3 | IC50 | 3 | — | |
XSHXVWHTZPAYJC
|
6.2 | Kd | 5 | — | |
YUNDLGQJZQUDNB
|
6.2 | IC50 | 4 | — | |
JZLPRLQRTFDCLM
|
6.2 | Kd | 4 | — | |
VXBVPENBQFGYRJ
|
6.1 | IC50 | 3 | — | |
VCAQDGBJOWAITH
|
6.1 | IC50 | 3 | — | |
DBUAWIKRKBNZMC
|
6.1 | Kd | 4 | — | |
SLIIQFIECPRWSD
|
6.1 | Kd | 3 | — |