Target Details
| UniProt AC | O00238 |
|---|---|
| Gene Symbol | BMPR1B |
| Protein Name | Bone morphogenetic protein receptor type-1B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF07714 (PK_Tyr_Ser-Thr) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 82
- Clinical molecules 12
- Avg pChEMBL 6.85
KEGG Pathways (7)
Associated Diseases (3)
Active Molecules (82)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VYPGLYMWNDRFGZ
|
6.5 | Kd | 12 | — | |
BLKUTJODYRMUJL
|
6.4 | IC50 | 4 | — | |
GUBJNPWVIUFSTR
|
6.4 | Kd | 103 | — | |
FYPPBYUPMODRPA
|
6.4 | IC50 | 4 | — | |
JOOXLOJCABQBSG
|
6.4 | Kd | 139 | — | |
UOAHJPVGHFVHGE
|
6.4 | IC50 | 4 | — | |
BIIVYFLTOXDAOV
|
6.3 | Kd | 82 | Yes | |
GGDVEPRDLUWBFD
|
6.3 | IC50 | 4 | — | |
OVNAOUBDNBHVCI
|
6.3 | IC50 | 5 | — | |
ITRDMWUZJMBHJF
|
6.3 | IC50 | 2 | — | |
QKDBOJCTMDJVMH
|
6.3 | IC50 | 4 | — | |
VMLFWTDHYNRGTR
|
6.3 | IC50 | 2 | — | |
ISWRGOFCPBCOGR
|
6.2 | IC50 | 3 | — | |
QYTUSJSFZCPMSV
|
6.2 | IC50 | 2 | — | |
MPVGZUGXCQEXTM
|
6.2 | Kd | 61 | Yes | |
HZMKNGJNPOBODV
|
6.1 | IC50 | 4 | — | |
IEJOMJUTRBOWNE
|
6.1 | Kd | 5 | — | |
NHHQJBCNYHBUSI
|
6.1 | Kd | 220 | — | |
QPIFMCLNACVAAT
|
6.1 | IC50 | 7 | — | |
PVDWNOWJXDXMDH
|
6.1 | IC50 | 5 | — | |
HIWHLPKRUZGHRR
|
6.1 | IC50 | 4 | — | |
QCXBJMRMYRQRCV
|
6.1 | IC50 | 4 | — | |
FCKKBQZIGVYODN
|
6.1 | IC50 | 4 | — | |
LJUBHCPBQBKBHM
|
6.0 | IC50 | 5 | — | |
CUIHSIWYWATEQL
|
6.0 | Kd | 61 | Yes | |
FZJGVHATMCAPLO
|
6.0 | IC50 | 5 | — | |
IFSNOUHZJMGMOD
|
6.0 | IC50 | 4 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
NTLWKKILBCETHV
|
6.0 | IC50 | 4 | — | |
ODVUZZFWFOPOAH
|
6.0 | IC50 | 5 | — |